Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50001450 ((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50016450 (CHEMBL39503 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50016451 (CHEMBL37306 | N-[2-(2-Amino-acetylamino)-ethyl]-2-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50226936 (CHEMBL37351) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50367270 (CHEMBL606297) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50367589 (CHEMBL3144091 | CHEMBL611126) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50226935 (CHEMBL3143947) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50226934 (CHEMBL3143946) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016446 (2-Amino-pentanedioic acid 5-amide 1-[(3-carbamoyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50367267 (CHEMBL605246) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50226934 (CHEMBL3143946) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016448 (2-Amino-pentanedioic acid 5-amide 1-({1-[1-({[1-(1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50367589 (CHEMBL3144091 | CHEMBL611126) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50367270 (CHEMBL606297) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016443 (2-{2-[2-(2-Acetylamino-3-phenyl-propionylamino)-3-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016445 (2-{2-[2-(2-Amino-3-phenyl-propionylamino)-3-phenyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016451 (CHEMBL37306 | N-[2-(2-Amino-acetylamino)-ethyl]-2-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50016450 (CHEMBL39503 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-P receptor (Rattus norvegicus (rat)) | BDBM50226935 (CHEMBL3143947) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slices | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50016443 (2-{2-[2-(2-Acetylamino-3-phenyl-propionylamino)-3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50001450 ((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1/A2a/A2b/A3 (Rattus norvegicus (rat)) | BDBM50016445 (2-{2-[2-(2-Amino-3-phenyl-propionylamino)-3-phenyl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranes | J Med Chem 30: 1529-32 (1987) BindingDB Entry DOI: 10.7270/Q24M954B | |||||||||||
More data for this Ligand-Target Pair |