Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50116661 (CHEMBL75668 | N-[(S)-1-(2,5-Dihydro-pyrrol-1-ylmet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Displacement of bound [3H]-diprenorphine in cloned rat Opioid receptor kappa 1 expressed in Sf9 insect cells | Bioorg Med Chem Lett 12: 2287-90 (2002) BindingDB Entry DOI: 10.7270/Q2QV3KTP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50116659 (2-(3,4-Dichloro-phenyl)-N-[(S)-1-(2,5-dihydro-pyrr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Displacement of bound [3H]-diprenorphine in cloned rat Opioid receptor kappa 1 expressed in Sf9 insect cells | Bioorg Med Chem Lett 12: 2287-90 (2002) BindingDB Entry DOI: 10.7270/Q2QV3KTP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539104 (CHEMBL4641260) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539105 (CHEMBL4636437) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539106 (CHEMBL4643799) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539107 (CHEMBL4639280) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539108 (CHEMBL4649247) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539109 (CHEMBL4634383) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539121 (CHEMBL4646130) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539111 (CHEMBL4646109) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539112 (CHEMBL4647600) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539113 (CHEMBL4649123) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539114 (CHEMBL4634892) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539115 (CHEMBL4635080) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539116 (CHEMBL4648147) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539117 (CHEMBL4648396) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539118 (CHEMBL4643228) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539119 (CHEMBL4635630) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539120 (CHEMBL4642813) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539103 (CHEMBL4636754) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539102 (CHEMBL7075) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Stress-70 protein, mitochondrial (Homo sapiens) | BDBM50539110 (CHEMBL4634635) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a |
Oklahoma State University Curated by ChEMBL | Assay Description Binding affinity to mortalin substrate binding domain (unknown origin) | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115244 BindingDB Entry DOI: 10.7270/Q2WD443B | |||||||||||
More data for this Ligand-Target Pair |