Found 2 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031319
(CHEMBL130853 | spiro[4,5-dihydro-1H-imidazole-4,2'...)Show InChI InChI=1S/C12H14N2/c1-2-4-11-7-12(8-13-9-14-12)6-5-10(11)3-1/h1-4,9H,5-8H2,(H,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Alpha-2B adrenergic receptor
(NEONATAL RAT) | BDBM50031319
(CHEMBL130853 | spiro[4,5-dihydro-1H-imidazole-4,2'...)Show InChI InChI=1S/C12H14N2/c1-2-4-11-7-12(8-13-9-14-12)6-5-10(11)3-1/h1-4,9H,5-8H2,(H,13,14) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 275 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2B adrenergic receptor in neonatal rat lung using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |