Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Melanocortin receptor 4
(Homo sapiens (Human)) | BDBM323223
(N-[(R)-1-(3,4-difluorobenzyl)-2-oxo-2-(3-pentyl-3-...)Show SMILES CCCCCC1(CN(C1)C(=O)[C@@H](Cc1ccc(F)c(F)c1)NC(=O)CCc1c[nH]cn1)c1ccccc1 Show InChI InChI=1S/C29H34F2N4O2/c1-2-3-7-14-29(22-8-5-4-6-9-22)18-35(19-29)28(37)26(16-21-10-12-24(30)25(31)15-21)34-27(36)13-11-23-17-32-20-33-23/h4-6,8-10,12,15,17,20,26H,2-3,7,11,13-14,16,18-19H2,1H3,(H,32,33)(H,34,36)/t26-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a |
GALDERMA RESEARCH & DEVELOPMENT
US Patent
| Assay Description
In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the... |
US Patent US9630949 (2017)
BindingDB Entry DOI: 10.7270/Q21Z46H9 |
More data for this
Ligand-Target Pair | |
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human)) | BDBM323223
(N-[(R)-1-(3,4-difluorobenzyl)-2-oxo-2-(3-pentyl-3-...)Show SMILES CCCCCC1(CN(C1)C(=O)[C@@H](Cc1ccc(F)c(F)c1)NC(=O)CCc1c[nH]cn1)c1ccccc1 Show InChI InChI=1S/C29H34F2N4O2/c1-2-3-7-14-29(22-8-5-4-6-9-22)18-35(19-29)28(37)26(16-21-10-12-24(30)25(31)15-21)34-27(36)13-11-23-17-32-20-33-23/h4-6,8-10,12,15,17,20,26H,2-3,7,11,13-14,16,18-19H2,1H3,(H,32,33)(H,34,36)/t26-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
GALDERMA RESEARCH & DEVELOPMENT
US Patent
| Assay Description
In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the... |
US Patent US9630949 (2017)
BindingDB Entry DOI: 10.7270/Q21Z46H9 |
More data for this
Ligand-Target Pair | |