Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Metabotropic glutamate receptor 3
(Rattus norvegicus (Rat)) | BDBM196832
(5-(4-fluorophenyl)-2-(((2-fluorophenyl)(methyl)ami...)Show SMILES CN(Cc1cc2C(=O)N(CCn2n1)c1ccc(F)cc1)c1ccccc1F Show InChI InChI=1S/C20H18F2N4O/c1-24(18-5-3-2-4-17(18)22)13-15-12-19-20(27)25(10-11-26(19)23-15)16-8-6-14(21)7-9-16/h2-9,12H,10-11,13H2,1H3 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 876 | n/a | n/a | n/a | n/a | n/a | 25 |
Vanderbilt University
US Patent
| Assay Description
HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m... |
US Patent US9676782 (2017)
BindingDB Entry DOI: 10.7270/Q2B8569W |
More data for this
Ligand-Target Pair | |
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat)) | BDBM196832
(5-(4-fluorophenyl)-2-(((2-fluorophenyl)(methyl)ami...)Show SMILES CN(Cc1cc2C(=O)N(CCn2n1)c1ccc(F)cc1)c1ccccc1F Show InChI InChI=1S/C20H18F2N4O/c1-24(18-5-3-2-4-17(18)22)13-15-12-19-20(27)25(10-11-26(19)23-15)16-8-6-14(21)7-9-16/h2-9,12H,10-11,13H2,1H3 | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | 25 |
Vanderbilt University
US Patent
| Assay Description
Gα15/TREx cells stably expressing rat mGlu3 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of a... |
US Patent US9676782 (2017)
BindingDB Entry DOI: 10.7270/Q2B8569W |
More data for this
Ligand-Target Pair | |