Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM274746
(N-(6-(4-(4-fluorophenyl)-1,2- dimethyl-1H-imidazol...)Show SMILES Cc1nc(c(-c2ccc3nc(NC(=O)c4ccc(O)nc4)cn3n2)n1C)-c1ccc(F)cc1 Show InChI InChI=1S/C23H18FN7O2/c1-13-26-21(14-3-6-16(24)7-4-14)22(30(13)2)17-8-9-19-27-18(12-31(19)29-17)28-23(33)15-5-10-20(32)25-11-15/h3-12H,1-2H3,(H,25,32)(H,28,33) | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 0.473 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |
Casein kinase I isoform epsilon
(Homo sapiens (Human)) | BDBM274746
(N-(6-(4-(4-fluorophenyl)-1,2- dimethyl-1H-imidazol...)Show SMILES Cc1nc(c(-c2ccc3nc(NC(=O)c4ccc(O)nc4)cn3n2)n1C)-c1ccc(F)cc1 Show InChI InChI=1S/C23H18FN7O2/c1-13-26-21(14-3-6-16(24)7-4-14)22(30(13)2)17-8-9-19-27-18(12-31(19)29-17)28-23(33)15-5-10-20(32)25-11-15/h3-12H,1-2H3,(H,25,32)(H,28,33) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 4.76 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |