Found 31 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Glutamate receptor 1
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
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| Article PubMed
| 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 1 (GluR1) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Rattus norvegicus (Rat)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[AMPA from rat recombinant GluA1o expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| Article PubMed
| 370 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[AMPA from rat recombinant GluA2(R)o expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
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| Article PubMed
| 370 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 2 (GluR2) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
KEGG
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| 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor ionotropic kainate 1 (GluR5) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 1
(RAT) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[SYM2081 from rat recombinant GluK1(Q)1b expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 4
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[AMPA from rat recombinant GluA4o expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 4
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 4 (GluR4) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 2C
(Rattus norvegicus (Rat)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined against N-methyl-D-aspartate glutamate receptor, using radioligand [3H]- CGP-39653 |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| 2.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[AMPA from rat recombinant GluA3o expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| 2.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor AMPA 3 (GluR3) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 3
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
KEGG
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| 9.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[SYM2081 from rat recombinant GluK3a expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 2
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined towards cloned Ionotropic glutamate receptor ionotropic kainate 6 (GluR6) expressed in Sf 9 insect cells |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 2
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Displacement of [3H[SYM2081 from rat recombinant GluK2(VCR)a expressed in sS9 cells |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Metabotropic glutamate receptor 1
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| Article PubMed
| 8.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Antagonist activity of compound at Metabotropic glutamate receptor 1 alpha was determined |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Rattus norvegicus (Rat)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| Article PubMed
| n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined against Ionotropic glutamate receptor AMPA receptor, using radioligand [3H]- AMPA |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, kainate 3
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
KEGG
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| Article PubMed
| n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Binding affinity of compound was determined against KA receptor,using radioligand [3H]- KA |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| Article PubMed
| n/a | n/a | n/a | n/a | 2.70E+6 | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Agonist activity at rat recombinant GluA3i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assay |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Agonist activity at rat recombinant GluA2(Q)i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assay |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Rattus norvegicus (Rat)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
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| Article PubMed
| n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Agonist activity at rat recombinant GluA1i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assay |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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| Article PubMed
| n/a | n/a | n/a | n/a | 2.70E+6 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at GluA3 receptor |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
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| Article PubMed
| n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at GluA2 receptor |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
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| Article PubMed
| n/a | n/a | n/a | n/a | 4.10E+3 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at GluA1 receptor |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
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Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 2.70E+6 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at recombinant GluA3 receptor flip isoform expressed in Xenopus oocytes |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |
Glutamate receptor 4
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
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Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 1.30E+6 | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Agonist activity at rat recombinant GluA4i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assay |
J Med Chem 53: 8354-8361 (2010)
Article DOI: 10.1021/jm101218a BindingDB Entry DOI: 10.7270/Q20Z73HW |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytes |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |
Glutamate receptor 3
(RAT) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 2.70E+6 | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 3 (GluR3) using rat cort... |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 4
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 1.30E+6 | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cort... |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Rattus norvegicus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 2 (GluR2) using rat cort... |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 1
(Mus musculus) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
The Danish University of Pharmaceutical Sciences
Curated by ChEMBL
| Assay Description Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 1 (GluR1) using rat cort... |
J Med Chem 46: 2246-9 (2003)
Article DOI: 10.1021/jm020588f BindingDB Entry DOI: 10.7270/Q26T0M06 |
More data for this Ligand-Target Pair | |
Glutamate receptor 2
(Homo sapiens (Human)) | BDBM50128264
((R,S)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)p...)Show InChI InChI=1S/C6H7ClN2O4/c7-4-3(13-9-5(4)10)1-2(8)6(11)12/h2H,1,8H2,(H,9,10)(H,11,12) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
University of California
Curated by ChEMBL
| Assay Description Agonist activity at recombinant GluA2 receptor flop isoform expressed in Xenopus oocytes |
Bioorg Med Chem 18: 1381-7 (2010)
Article DOI: 10.1016/j.bmc.2009.12.072 BindingDB Entry DOI: 10.7270/Q27W6CB2 |
More data for this Ligand-Target Pair | |