Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Dipeptidyl peptidase 1
(Homo sapiens (Human)) | BDBM153533
(BDBM153612 | US8999975, 50)Show SMILES O[C@H]1C[C@H]2C[C@@H]1N[C@@H]2C(=O)N[C@@H](Cc1ccc(cc1)-c1ccc(C#N)c(F)c1)C#N |r| Show InChI InChI=1S/C23H21FN4O2/c24-19-8-15(5-6-16(19)11-25)14-3-1-13(2-4-14)7-18(12-26)27-23(30)22-17-9-20(28-22)21(29)10-17/h1-6,8,17-18,20-22,28-29H,7,9-10H2,(H,27,30)/t17-,18+,20+,21+,22+/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
Similars
| US Patent
| n/a | n/a | 13 | n/a | n/a | n/a | n/a | 6.0 | 25 |
Boehringer Ingelheim International GmbH
US Patent
| Assay Description
The following buffers were used: MES buffer: 25 mM MES, 50 mM NaCl, 5 mM DTT, adjusted to pH 6.0, containing 0.1% BSA; TAGZyme Buffer: 20 mM NaH2PO4,... |
US Patent US8999975 (2015)
BindingDB Entry DOI: 10.7270/Q22806BZ |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 1
(Homo sapiens (Human)) | BDBM153533
(BDBM153612 | US8999975, 50)Show SMILES O[C@H]1C[C@H]2C[C@@H]1N[C@@H]2C(=O)N[C@@H](Cc1ccc(cc1)-c1ccc(C#N)c(F)c1)C#N |r| Show InChI InChI=1S/C23H21FN4O2/c24-19-8-15(5-6-16(19)11-25)14-3-1-13(2-4-14)7-18(12-26)27-23(30)22-17-9-20(28-22)21(29)10-17/h1-6,8,17-18,20-22,28-29H,7,9-10H2,(H,27,30)/t17-,18+,20+,21+,22+/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
Similars
| US Patent
| n/a | n/a | 14 | n/a | n/a | n/a | n/a | 6.0 | 25 |
Boehringer Ingelheim International GmbH
US Patent
| Assay Description
The following buffers were used: MES buffer: 25 mM MES, 50 mM NaCl, 5 mM DTT, adjusted to pH 6.0, containing 0.1% BSA; TAGZyme Buffer: 20 mM NaH2PO4,... |
US Patent US8999975 (2015)
BindingDB Entry DOI: 10.7270/Q22806BZ |
More data for this
Ligand-Target Pair | |