Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Lysophosphatidic acid receptor 1
(Homo sapiens (Human)) | BDBM251719
(US10100018, Example 55 | US9464060, 55)Show SMILES OC(=O)c1ccc(CN(Cc2ccccc2)C(=O)C2CCC(CC2)Oc2ccccc2F)cc1 |(7.34,-5.77,;7.34,-4.24,;8.67,-3.47,;6,-3.47,;4.67,-4.24,;3.33,-3.47,;3.33,-1.93,;2,-1.16,;2,.38,;3.33,1.15,;3.33,2.69,;4.67,3.46,;4.67,5,;3.33,5.77,;2,5,;2,3.46,;.67,1.15,;.67,2.69,;-.67,.38,;-2,1.15,;-3.33,.38,;-3.33,-1.16,;-2,-1.93,;-.67,-1.16,;-4.67,-1.93,;-6,-1.16,;-6,.38,;-7.34,1.15,;-8.67,.38,;-8.67,-1.16,;-7.34,-1.93,;-7.34,-3.46,;4.67,-1.16,;6,-1.93,)| Show InChI InChI=1S/C28H28FNO4/c29-25-8-4-5-9-26(25)34-24-16-14-22(15-17-24)27(31)30(18-20-6-2-1-3-7-20)19-21-10-12-23(13-11-21)28(32)33/h1-13,22,24H,14-19H2,(H,32,33) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | 25 |
Takeda Pharmaceutical Company Limited
US Patent
| Assay Description
Engagement of the LPA1 receptor by its ligand, oleoyl-L-α-lysophosphatidic acid (LPA), leads to the release of intracellular stores of calcium i... |
US Patent US10100018 (2018)
BindingDB Entry DOI: 10.7270/Q2PR7Z0N |
More data for this
Ligand-Target Pair | |
Lysophosphatidic acid receptor 5
(Homo sapiens (Human)) | BDBM251719
(US10100018, Example 55 | US9464060, 55)Show SMILES OC(=O)c1ccc(CN(Cc2ccccc2)C(=O)C2CCC(CC2)Oc2ccccc2F)cc1 |(7.34,-5.77,;7.34,-4.24,;8.67,-3.47,;6,-3.47,;4.67,-4.24,;3.33,-3.47,;3.33,-1.93,;2,-1.16,;2,.38,;3.33,1.15,;3.33,2.69,;4.67,3.46,;4.67,5,;3.33,5.77,;2,5,;2,3.46,;.67,1.15,;.67,2.69,;-.67,.38,;-2,1.15,;-3.33,.38,;-3.33,-1.16,;-2,-1.93,;-.67,-1.16,;-4.67,-1.93,;-6,-1.16,;-6,.38,;-7.34,1.15,;-8.67,.38,;-8.67,-1.16,;-7.34,-1.93,;-7.34,-3.46,;4.67,-1.16,;6,-1.93,)| Show InChI InChI=1S/C28H28FNO4/c29-25-8-4-5-9-26(25)34-24-16-14-22(15-17-24)27(31)30(18-20-6-2-1-3-7-20)19-21-10-12-23(13-11-21)28(32)33/h1-13,22,24H,14-19H2,(H,32,33) | UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | 37 |
Takeda Pharmaceutical Company Limited
US Patent
| Assay Description
Engagement of the LPA5 receptor by its ligand, oleoyl-L-α-lysophosphatidic acid (LPA), leads to the release of intracellular stores of calcium into ... |
US Patent US9464060 (2016)
BindingDB Entry DOI: 10.7270/Q23R0RT0 |
More data for this
Ligand-Target Pair | |