Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Formyl peptide receptor 2 (Mus musculus) | BDBM50559829 (CHEMBL4784510) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559829 (CHEMBL4784510) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | <1 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at FPR2 in mouse peritoneal macrophages assessed as inhibition of stimulated phagocytosis preincubated for 15 mins followed by FITC ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559821 (CHEMBL4781596) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559829 (CHEMBL4784510) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559829 (CHEMBL4784510) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | n/a | n/a | n/a | n/a | 384 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559838 (CHEMBL4790836) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.630 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559840 (CHEMBL4760897) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50186957 (1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Formyl peptide receptor 2 (Mus musculus) | BDBM50559835 (CHEMBL4762030) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni... | Citation and Details Article DOI: 10.1021/acs.jmedchem.9b02101 BindingDB Entry DOI: 10.7270/Q2V98CSC | |||||||||||
More data for this Ligand-Target Pair |