Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50514481 (CHEMBL3782104) | UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Zambia Curated by ChEMBL | Assay Description Inhibition of recombinant Plasmodium falciparum Plasmepsin 5 | J Med Chem 63: 4445-4467 (2020) Article DOI: 10.1021/acs.jmedchem.9b01622 BindingDB Entry DOI: 10.7270/Q2RR22K7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50500851 (CHEMBL3780033) | UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Melbourne Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum PMV assessed as fluorogenic substrate cleavage using DABCYL-RNKRTLAQKQ-E-EDANS as fluorogenic substrate after 120... | Bioorg Med Chem 24: 1993-2010 (2016) Article DOI: 10.1016/j.bmc.2016.03.027 BindingDB Entry DOI: 10.7270/Q21R6THF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099406 (CHEMBL3344272) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium vivax) | BDBM50099406 (CHEMBL3344272) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium vivax plasmepsin V by fluorogenic PEXEL cleavage assay | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099378 (CHEMBL3344165) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099272 (CHEMBL3344164) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099380 (CHEMBL3344166) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 77 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099381 (CHEMBL3344261) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099391 (CHEMBL3344266) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 348 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099395 (CHEMBL3344270) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 378 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099387 (CHEMBL3344262) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099394 (CHEMBL3344269) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099148 (CHEMBL3344151) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 556 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099390 (CHEMBL3344265) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 569 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099171 (CHEMBL3344152) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 613 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099240 (CHEMBL3344157) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 614 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099388 (CHEMBL3344263) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 622 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099403 (CHEMBL3344271) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 625 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099389 (CHEMBL3344264) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 772 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099393 (CHEMBL3344268) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 774 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099236 (CHEMBL3344153) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 865 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099237 (CHEMBL3344154) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 967 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099392 (CHEMBL3344267) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099239 (CHEMBL3344156) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099238 (CHEMBL3344155) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099242 (CHEMBL3344159) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099241 (CHEMBL3344158) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099247 (CHEMBL3344161) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099249 (CHEMBL3344162) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099252 (CHEMBL3344163) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasmepsin V (Plasmodium falciparum (isolate 3D7)) | BDBM50099243 (CHEMBL3344160) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrate | J Med Chem 57: 7644-62 (2014) Article DOI: 10.1021/jm500797g BindingDB Entry DOI: 10.7270/Q2CR5W42 | |||||||||||
More data for this Ligand-Target Pair |