Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein lifeguard 1 (BOVINE) | BDBM86757 (CAS_0 | NSC_11603174 | [11C]MMP) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Columbia University Curated by PDSP Ki Database | Eur J Nucl Med Mol Imaging 34: 1050-60 (2007) Article DOI: 10.1007/s00259-006-0324-y BindingDB Entry DOI: 10.7270/Q2D7990W | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein lifeguard 1 (Rattus norvegicus) | BDBM50118479 (2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.87E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Binding affinity towards N-methyl-D-aspartate glutamate receptor (NMDA) determined electrophysically using the rat cortical wedge model. | J Med Chem 45: 4240-5 (2002) BindingDB Entry DOI: 10.7270/Q28G8K2W | |||||||||||
More data for this Ligand-Target Pair |