Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200114 (CHEMBL3920498) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.86E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assay | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200114 (CHEMBL3920498) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assay | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200111 (CHEMBL3981566) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 9.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assay | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200111 (CHEMBL3981566) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 3.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assay | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50548078 (CHEMBL4746798) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0280 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524090 (6-{[3-(2-Fluoropyridin-3-yl)-1H-pyrazol-1-yl]methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0340 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524080 (6-{[3-(2-Fluorophenyl)-1H-pyrazol-1-yl]methyl}-5-m...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524098 (US11136337, Example 4.9) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524101 (US11136337, Example 4.12) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0760 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524097 (US11136337, Example 4.8) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.0960 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524091 (US11136337, Example 4.2) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524092 (US11136337, Example 4.3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524099 (US11136337, Example 4.10) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524095 (US11136337, Example 4.6) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524084 (US11136337, Example 2.5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524100 (US11136337, Example 4.11) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524103 (US11136337, Example 4.14) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524081 (US11136337, Example 2.2) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524082 (US11136337, Example 2.3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524093 (US11136337, Example 4.4) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.290 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524096 (US11136337, Example 4.7) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.370 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524102 (US11136337, Example 4.13) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524074 (US11136337, Example 1.4) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.510 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524077 (US11136337, Example 1.7) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524107 (6-[(2H-Indazol-2-yl)methyl]-5-methyl-[1,2,5]oxadia...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.690 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524108 (6-{[3-(3,3-Difluoropyrrolidine-1-carbonyl)-1H-pyra...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.840 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524076 (US11136337, Example 1.6) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524087 (US11136337, Example 3.2) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524078 (US11136337, Example 1.8) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524072 (US11136337, Example 1.2) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524083 (US11136337, Example 2.4) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524071 (Ethyl 1-({7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524073 (US11136337, Example 1.3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524088 (US11136337, Example 3.3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524111 (Benzyl N-(1-{[1-({7-amino-5-methyl-[1,2,5]oxadiazo...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524075 (US11136337, Example 1.5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524086 (1.1 6-{[4-(3-Methanesulfonylphenyl)-3-(trifluorome...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524109 (US11136337, Example 7.2) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524105 (US11136337, Example 4.16) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524094 (US11136337, Example 4.5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524085 (US11136337, Example 2.6) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524079 (US11136337, Example 1.9) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524110 (US11136337, Example 7.3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524089 (US11136337, Example 3.4) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524104 (US11136337, Example 4.15) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM524112 (6-({3-[(4,4-Difluoropiperidin-1-yl)methyl]-1H-pyra...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Each assay plate contains wells with vehicle controls (1% DMSO) for the measurement of non-inhibited transfer reaction (=100% Ctl) and wells with 10 ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2028VQ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50118239 (CHEMBL130266 | UDP | Uridine diphosphate | uridine...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of British Columbia Curated by ChEMBL | Assay Description Inhibition of human OGT | Bioorg Med Chem Lett 21: 1199-201 (2011) Article DOI: 10.1016/j.bmcl.2010.12.090 BindingDB Entry DOI: 10.7270/Q2028RT6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50168000 (3H-Benzooxazol-2-one | CHEMBL280323 | benzo[d]oxaz...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC method | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200114 (CHEMBL3920498) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.67E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC method | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit (Homo sapiens (Human)) | BDBM50200110 (CHEMBL3890166) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Chinese Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC method | J Med Chem 60: 263-272 (2017) Article DOI: 10.1021/acs.jmedchem.6b01237 BindingDB Entry DOI: 10.7270/Q20G3N47 | |||||||||||
More data for this Ligand-Target Pair |
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