Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263227 (US9708370, GHRP-6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 3.65 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263217 (US9708370, DBG-253-10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 465 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263226 (US9708370, DBG-168-8p) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 514 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394997 (CHEMBL2163482 | US9708370, DBG-253-6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 723 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263218 (US9708370, DBG-253-11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 729 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394996 (CHEMBL2163348 | US9708370, DBG-253-7) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 771 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50395003 (CHEMBL2163476 | US9708370, DBG-188p) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 808 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263225 (US9708370, DBG-145p) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 809 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50395002 (CHEMBL2163477 | US9708370, DBG-201-A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394999 (CHEMBL2163480 | US9708370, DBG-253-3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.34E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263219 (US9708370, DBG-253-12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.64E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50395001 (CHEMBL2163478 | US9708370, DBG-253-1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 2.77E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394995 (CHEMBL2163483 | US9708370, DBG-253-8) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 3.25E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394998 (CHEMBL2163481 | US9708370, DBG-253-5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 3.74E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM254027 (US9708370, DBG-253-4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 4.28E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263220 (US9708370, DBG-253-13) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 5.49E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263222 (US9708370, DBG-175p) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 8.53E+3 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50394994 (CHEMBL2163484 | US9708370, DBG-178p) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.57E+4 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM263216 (US9708370, DBG-253-9) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.61E+4 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [D538G] (Homo sapiens (Human)) | BDBM50395000 (CHEMBL2163479 | US9708370, DBG-253-2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | n/a | n/a | 1.95E+4 | n/a | n/a | n/a | n/a |
VALORISATION-RECHERCHE, LIMITED PARTNERSHIP; VALORISATION HSJ, LIMITED PARTNERSHIP US Patent | Assay Description GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer. | US Patent US9708370 (2017) BindingDB Entry DOI: 10.7270/Q2XP76ZK | |||||||||||
More data for this Ligand-Target Pair |