Compile Data Set for Download or QSAR

Found 458 hits of ic50 for UniProtKB: P30530   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298989 (US10125118, Example 395 | US10947215, Example 395) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccncc2)ccc1C |r| Show InChI InChI=1S/C25H29N5O2/c1-3-18-10-17(5-4-16(18)2)15-32-23-14-28-13-22(23)30-25(31)21-11-20(12-29-24(21)26)19-6-8-27-9-7-19/h4-12,22-23,28H,3,13-15H2,1-2H3,(H2,26,29)(H,30,31)/t22-,23-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298990 (US10125118, Example 396 | US10947215, Example 396) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cccnc2)ccc1C |r| Show InChI InChI=1S/C25H29N5O2/c1-3-18-9-17(7-6-16(18)2)15-32-23-14-28-13-22(23)30-25(31)21-10-20(12-29-24(21)26)19-5-4-8-27-11-19/h4-12,22-23,28H,3,13-15H2,1-2H3,(H2,26,29)(H,30,31)/t22-,23-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298993 (US10125118, Example 399 | US10947215, Example 399) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(OC)cc2)ccc1C |r| Show InChI InChI=1S/C27H32N4O3/c1-4-19-11-18(6-5-17(19)2)16-34-25-15-29-14-24(25)31-27(32)23-12-21(13-30-26(23)28)20-7-9-22(33-3)10-8-20/h5-13,24-25,29H,4,14-16H2,1-3H3,(H2,28,30)(H,31,32)/t24-,25-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM486769 (US10947215, Example 400) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(cc2)C#N)ccc1C |r| Show InChI InChI=1S/C27H29N5O2/c1-3-20-10-19(5-4-17(20)2)16-34-25-15-30-14-24(25)32-27(33)23-11-22(13-31-26(23)29)21-8-6-18(12-28)7-9-21/h4-11,13,24-25,30H,3,14-16H2,1-2H3,(H2,29,31)(H,32,33)/t24-,25-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298995 (US10125118, Example 401 | US10947215, Example 401) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(NS(C)(=O)=O)cc2)ccc1C |r| Show InChI InChI=1S/C27H33N5O4S/c1-4-19-11-18(6-5-17(19)2)16-36-25-15-29-14-24(25)31-27(33)23-12-21(13-30-26(23)28)20-7-9-22(10-8-20)32-37(3,34)35/h5-13,24-25,29,32H,4,14-16H2,1-3H3,(H2,28,30)(H,31,33)/t24-,25-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298999 (US10125118, Example 405 | US10947215, Example 405) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(cc2)N(C)C)ccc1C |r| Show InChI InChI=1S/C28H35N5O2/c1-5-20-12-19(7-6-18(20)2)17-35-26-16-30-15-25(26)32-28(34)24-13-22(14-31-27(24)29)21-8-10-23(11-9-21)33(3)4/h6-14,25-26,30H,5,15-17H2,1-4H3,(H2,29,31)(H,32,34)/t25-,26-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM486780 (US10947215, Example 411) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(CC#N)cc2)ccc1C |r| Show InChI InChI=1S/C28H31N5O2/c1-3-21-12-20(5-4-18(21)2)17-35-26-16-31-15-25(26)33-28(34)24-13-23(14-32-27(24)30)22-8-6-19(7-9-22)10-11-29/h4-9,12-14,25-26,31H,3,10,15-17H2,1-2H3,(H2,30,32)(H,33,34)/t25-,26-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299006 (US10125118, Example 412 | US10947215, Example 412) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(c2)C2CCNCC2)ccc1C |r| Show InChI InChI=1S/C28H37N7O2/c1-3-20-10-19(5-4-18(20)2)17-37-26-15-31-14-25(26)34-28(36)24-11-21(12-32-27(24)29)22-13-33-35(16-22)23-6-8-30-9-7-23/h4-5,10-13,16,23,25-26,30-31H,3,6-9,14-15,17H2,1-2H3,(H2,29,32)(H,34,36)/t25-,26-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299007 (US10125118, Example 413 | US10947215, Example 413) Show SMILES CCc1cc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(c2)C2CCN(C)CC2)ccc1C |r| Show InChI InChI=1S/C29H39N7O2/c1-4-21-11-20(6-5-19(21)2)18-38-27-16-31-15-26(27)34-29(37)25-12-22(13-32-28(25)30)23-14-33-36(17-23)24-7-9-35(3)10-8-24/h5-6,11-14,17,24,26-27,31H,4,7-10,15-16,18H2,1-3H3,(H2,30,32)(H,34,37)/t26-,27-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299009 (US10125118, Example 415 | US10947215, Example 415) Show SMILES Cc1ccc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C22H26N6O2/c1-14-3-5-15(6-4-14)13-30-20-11-24-10-19(20)27-22(29)18-7-16(8-25-21(18)23)17-9-26-28(2)12-17/h3-9,12,19-20,24H,10-11,13H2,1-2H3,(H2,23,25)(H,27,29)/t19-,20-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299010 (US10125118, Example 416 | US10947215, Example 416) Show SMILES CCc1cccc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)c1 |r| Show InChI InChI=1S/C23H28N6O2/c1-3-15-5-4-6-16(7-15)14-31-21-12-25-11-20(21)28-23(30)19-8-17(9-26-22(19)24)18-10-27-29(2)13-18/h4-10,13,20-21,25H,3,11-12,14H2,1-2H3,(H2,24,26)(H,28,30)/t20-,21-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM486788 (US10947215, Example 419) Show SMILES CCc1cc(CO[C@H]2CN(C[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(cc2)C(O)=O)C(=O)OC(C)(C)C)ccc1C |r| Show InChI InChI=1S/C32H38N4O6/c1-6-21-13-20(8-7-19(21)2)18-41-27-17-36(31(40)42-32(3,4)5)16-26(27)35-29(37)25-14-24(15-34-28(25)33)22-9-11-23(12-10-22)30(38)39/h7-15,26-27H,6,16-18H2,1-5H3,(H2,33,34)(H,35,37)(H,38,39)/t26-,27-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299020 (US10125118, Example 426 | US10125118, Example 433 ...) Show SMILES CCc1cc(CO[C@H]2CN(C)C[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)ccc1C |r| Show InChI InChI=1S/C25H32N6O2/c1-5-18-8-17(7-6-16(18)2)15-33-23-14-30(3)13-22(23)29-25(32)21-9-19(10-27-24(21)26)20-11-28-31(4)12-20/h6-12,22-23H,5,13-15H2,1-4H3,(H2,26,27)(H,29,32)/t22-,23-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM486802 (US10947215, Example 433) Show SMILES CCc1cc(CO[C@H]2CN(C)C[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(c2)C2CCN(C)CC2)ccc1C |r| Show InChI InChI=1S/C30H41N7O2/c1-5-22-12-21(7-6-20(22)2)19-39-28-18-36(4)17-27(28)34-30(38)26-13-23(14-32-29(26)31)24-15-33-37(16-24)25-8-10-35(3)11-9-25/h6-7,12-16,25,27-28H,5,8-11,17-19H2,1-4H3,(H2,31,32)(H,34,38)/t27-,28-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299028 (US10125118, Example 434 | US10947215, Example 434) Show SMILES CN1CCN(Cc2ccc(cc2)-c2ccc(CO[C@H]3CNC[C@@H]3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C33H40N8O2/c1-39-11-13-41(14-12-39)20-23-3-7-25(8-4-23)26-9-5-24(6-10-26)22-43-31-19-35-18-30(31)38-33(42)29-15-27(16-36-32(29)34)28-17-37-40(2)21-28/h3-10,15-17,21,30-31,35H,11-14,18-20,22H2,1-2H3,(H2,34,36)(H,38,42)/t30-,31-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299029 (US10125118, Example 435 | US10947215, Example 435) Show SMILES CN1C[C@H](NC(=O)c2cc(cnc2N)-c2cnn(C)c2)[C@H](C1)OCc1ccc(cc1)-c1ccc(CN2CCN(C)CC2)cc1 |r| Show InChI InChI=1S/C34H42N8O2/c1-39-12-14-42(15-13-39)19-24-4-8-26(9-5-24)27-10-6-25(7-11-27)23-44-32-22-40(2)21-31(32)38-34(43)30-16-28(17-36-33(30)35)29-18-37-41(3)20-29/h4-11,16-18,20,31-32H,12-15,19,21-23H2,1-3H3,(H2,35,36)(H,38,43)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299030 (US10125118, Example 436 | US10947215, Example 436) Show SMILES CN1CCN(Cc2ccc(cc2C(F)(F)F)-c2ccc(CO[C@H]3CNC[C@@H]3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C34H39F3N8O2/c1-43-9-11-45(12-10-43)20-25-8-7-24(14-29(25)34(35,36)37)23-5-3-22(4-6-23)21-47-31-18-39-17-30(31)42-33(46)28-13-26(15-40-32(28)38)27-16-41-44(2)19-27/h3-8,13-16,19,30-31,39H,9-12,17-18,20-21H2,1-2H3,(H2,38,40)(H,42,46)/t30-,31-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299031 (US10125118, Example 437 | US10947215, Example 437) Show SMILES CN1C[C@H](NC(=O)c2cc(cnc2N)-c2cnn(C)c2)[C@H](C1)OCc1ccc(cc1)-c1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F |r| Show InChI InChI=1S/C35H41F3N8O2/c1-43-10-12-46(13-11-43)19-26-9-8-25(15-30(26)35(36,37)38)24-6-4-23(5-7-24)22-48-32-21-44(2)20-31(32)42-34(47)29-14-27(16-40-33(29)39)28-17-41-45(3)18-28/h4-9,14-18,31-32H,10-13,19-22H2,1-3H3,(H2,39,40)(H,42,47)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299032 (US10125118, Example 438 | US10947215, Example 438) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C34H42N8O2/c1-23(42-14-12-40(2)13-15-42)25-8-10-27(11-9-25)26-6-4-24(5-7-26)22-44-32-20-36-19-31(32)39-34(43)30-16-28(17-37-33(30)35)29-18-38-41(3)21-29/h4-11,16-18,21,23,31-32,36H,12-15,19-20,22H2,1-3H3,(H2,35,37)(H,39,43)/t23?,31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299033 (US10125118, Example 439 | US10947215, Example 439) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CN(C)C[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C35H44N8O2/c1-24(43-15-13-40(2)14-16-43)26-9-11-28(12-10-26)27-7-5-25(6-8-27)23-45-33-22-41(3)21-32(33)39-35(44)31-17-29(18-37-34(31)36)30-19-38-42(4)20-30/h5-12,17-20,24,32-33H,13-16,21-23H2,1-4H3,(H2,36,37)(H,39,44)/t24?,32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299034 (US10125118, Example 440 | US10947215, Example 440) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1CNC[C@@H]1OCc1ccc(cc1)-c1ccc(cc1)C(C)(C)N1CCN(CCO)CC1 |r| Show InChI InChI=1S/C36H46N8O3/c1-36(2,44-14-12-43(13-15-44)16-17-45)30-10-8-27(9-11-30)26-6-4-25(5-7-26)24-47-33-22-38-21-32(33)41-35(46)31-18-28(19-39-34(31)37)29-20-40-42(3)23-29/h4-11,18-20,23,32-33,38,45H,12-17,21-22,24H2,1-3H3,(H2,37,39)(H,41,46)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299035 (US10125118, Example 441 | US10947215, Example 441) Show SMILES CN1C[C@H](NC(=O)c2cc(cnc2N)-c2cnn(C)c2)[C@H](C1)OCc1ccc(cc1)-c1ccc(cc1)C(C)(C)N1CCN(CCO)CC1 |r| Show InChI InChI=1S/C37H48N8O3/c1-37(2,45-15-13-44(14-16-45)17-18-46)31-11-9-28(10-12-31)27-7-5-26(6-8-27)25-48-34-24-42(3)23-33(34)41-36(47)32-19-29(20-39-35(32)38)30-21-40-43(4)22-30/h5-12,19-22,33-34,46H,13-18,23-25H2,1-4H3,(H2,38,39)(H,41,47)/t33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299036 (US10125118, Example 442 | US10947215, Example 442) Show SMILES CC(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CNC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C35H44N8O3/c1-24(43-13-11-42(12-14-43)15-16-44)26-7-9-28(10-8-26)27-5-3-25(4-6-27)23-46-33-21-37-20-32(33)40-35(45)31-17-29(18-38-34(31)36)30-19-39-41(2)22-30/h3-10,17-19,22,24,32-33,37,44H,11-16,20-21,23H2,1-2H3,(H2,36,38)(H,40,45)/t24?,32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299037 (US10125118, Example 443 | US10947215, Example 443) Show SMILES CC(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CN(C)C[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C36H46N8O3/c1-25(44-14-12-43(13-15-44)16-17-45)27-8-10-29(11-9-27)28-6-4-26(5-7-28)24-47-34-23-41(2)22-33(34)40-36(46)32-18-30(19-38-35(32)37)31-20-39-42(3)21-31/h4-11,18-21,25,33-34,45H,12-17,22-24H2,1-3H3,(H2,37,38)(H,40,46)/t25?,33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299038 (US10125118, Example 444 | US10947215, Example 444) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1CNC[C@@H]1OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F |r| Show InChI InChI=1S/C35H41F3N8O3/c1-44-20-28(17-42-44)27-14-29(33(39)41-16-27)34(48)43-31-18-40-19-32(31)49-22-23-2-4-24(5-3-23)25-6-7-26(30(15-25)35(36,37)38)21-46-10-8-45(9-11-46)12-13-47/h2-7,14-17,20,31-32,40,47H,8-13,18-19,21-22H2,1H3,(H2,39,41)(H,43,48)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299039 (US10125118, Example 445 | US10947215, Example 445) Show SMILES CN1C[C@H](NC(=O)c2cc(cnc2N)-c2cnn(C)c2)[C@H](C1)OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F |r| Show InChI InChI=1S/C36H43F3N8O3/c1-44-21-32(43-35(49)30-15-28(17-41-34(30)40)29-18-42-45(2)19-29)33(22-44)50-23-24-3-5-25(6-4-24)26-7-8-27(31(16-26)36(37,38)39)20-47-11-9-46(10-12-47)13-14-48/h3-8,15-19,32-33,48H,9-14,20-23H2,1-2H3,(H2,40,41)(H,43,49)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299040 (US10125118, Example 446 | US10947215, Example 446) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1CNC[C@@H]1OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)cc1 |r| Show InChI InChI=1S/C34H42N8O3/c1-40-22-29(18-38-40)28-16-30(33(35)37-17-28)34(44)39-31-19-36-20-32(31)45-23-25-4-8-27(9-5-25)26-6-2-24(3-7-26)21-42-12-10-41(11-13-42)14-15-43/h2-9,16-18,22,31-32,36,43H,10-15,19-21,23H2,1H3,(H2,35,37)(H,39,44)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299041 (US10125118, Example 447 | US10947215, Example 447) Show SMILES CN1C[C@H](NC(=O)c2cc(cnc2N)-c2cnn(C)c2)[C@H](C1)OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)cc1 |r| Show InChI InChI=1S/C35H44N8O3/c1-40-22-32(39-35(45)31-17-29(18-37-34(31)36)30-19-38-41(2)21-30)33(23-40)46-24-26-5-9-28(10-6-26)27-7-3-25(4-8-27)20-43-13-11-42(12-14-43)15-16-44/h3-10,17-19,21,32-33,44H,11-16,20,22-24H2,1-2H3,(H2,36,37)(H,39,45)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299042 (US10125118, Example 448 | US10947215, Example 448) Show SMILES CN1CCN(Cc2ccc(cc2)-c2ccc(CO[C@H]3COC[C@@H]3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C33H39N7O3/c1-38-11-13-40(14-12-38)18-23-3-7-25(8-4-23)26-9-5-24(6-10-26)20-43-31-22-42-21-30(31)37-33(41)29-15-27(16-35-32(29)34)28-17-36-39(2)19-28/h3-10,15-17,19,30-31H,11-14,18,20-22H2,1-2H3,(H2,34,35)(H,37,41)/t30-,31-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299043 (US10125118, Example 449 | US10947215, Example 449) Show SMILES CN1CCN(Cc2ccc(cc2C(F)(F)F)-c2ccc(CO[C@H]3COC[C@@H]3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C34H38F3N7O3/c1-42-9-11-44(12-10-42)18-25-8-7-24(14-29(25)34(35,36)37)23-5-3-22(4-6-23)19-47-31-21-46-20-30(31)41-33(45)28-13-26(15-39-32(28)38)27-16-40-43(2)17-27/h3-8,13-17,30-31H,9-12,18-21H2,1-2H3,(H2,38,39)(H,41,45)/t30-,31-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299044 (US10125118, Example 450 | US10947215, Example 450) Show SMILES CN1CCN(CC1)C(C)(C)c1ccc(cc1)-c1ccc(CO[C@H]2COC[C@@H]2NC(=O)c2cc(cnc2N)-c2cnn(C)c2)cc1 |r| Show InChI InChI=1S/C35H43N7O3/c1-35(2,42-15-13-40(3)14-16-42)29-11-9-26(10-12-29)25-7-5-24(6-8-25)21-45-32-23-44-22-31(32)39-34(43)30-17-27(18-37-33(30)36)28-19-38-41(4)20-28/h5-12,17-20,31-32H,13-16,21-23H2,1-4H3,(H2,36,37)(H,39,43)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299045 (US10125118, Example 451 | US10947215, Example 451) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1COC[C@@H]1OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)cc1 |r| Show InChI InChI=1S/C34H41N7O4/c1-39-20-29(18-37-39)28-16-30(33(35)36-17-28)34(43)38-31-22-44-23-32(31)45-21-25-4-8-27(9-5-25)26-6-2-24(3-7-26)19-41-12-10-40(11-13-41)14-15-42/h2-9,16-18,20,31-32,42H,10-15,19,21-23H2,1H3,(H2,35,36)(H,38,43)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299046 (US10125118, Example 452 | US10947215, Example 452) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1COC[C@@H]1OCc1ccc(cc1)-c1ccc(CN2CCN(CCO)CC2)c(c1)C(F)(F)F |r| Show InChI InChI=1S/C35H40F3N7O4/c1-43-18-28(17-41-43)27-14-29(33(39)40-16-27)34(47)42-31-21-48-22-32(31)49-20-23-2-4-24(5-3-23)25-6-7-26(30(15-25)35(36,37)38)19-45-10-8-44(9-11-45)12-13-46/h2-7,14-18,31-32,46H,8-13,19-22H2,1H3,(H2,39,40)(H,42,47)/t31-,32-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299047 (US10125118, Example 453 | US10947215, Example 453) Show SMILES Cn1cc(cn1)-c1cnc(N)c(c1)C(=O)N[C@H]1COC[C@@H]1OCc1ccc(cc1)-c1ccc(cc1)C(C)(C)N1CCN(CCO)CC1 |r| Show InChI InChI=1S/C36H45N7O4/c1-36(2,43-14-12-42(13-15-43)16-17-44)30-10-8-27(9-11-30)26-6-4-25(5-7-26)22-47-33-24-46-23-32(33)40-35(45)31-18-28(19-38-34(31)37)29-20-39-41(3)21-29/h4-11,18-21,32-33,44H,12-17,22-24H2,1-3H3,(H2,37,38)(H,40,45)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM299048 (US10125118, Example 454 | US10947215, Example 454) Show SMILES CN1CCN(Cc2ccc(cc2)-c2ccc(CO[C@H]3COCC3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C33H39N7O3/c1-38-11-13-40(14-12-38)18-23-3-7-25(8-4-23)26-9-5-24(6-10-26)20-43-31-22-42-21-30(31)37-33(41)29-15-27(16-35-32(29)34)28-17-36-39(2)19-28/h3-10,15-17,19,30-31H,11-14,18,20-22H2,1-2H3,(H2,34,35)(H,37,41)/t30?,31-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298818 (US10125118, Example 224 | US10947215, Example 224) Show SMILES CN1CCN(CC1)C1(CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C37H41FN6O2/c1-43-17-19-44(20-18-43)37(15-16-37)30-12-9-27(10-13-30)26-7-5-25(6-8-26)24-46-33-4-2-3-32(33)42-36(45)31-21-29(23-41-35(31)39)28-11-14-34(38)40-22-28/h5-14,21-23,32-33H,2-4,15-20,24H2,1H3,(H2,39,41)(H,42,45)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298819 (US10125118, Example 225 | US10947215, Example 225) Show SMILES CN1CCN(CC1)C(C)(C)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C37H43FN6O2/c1-37(2,44-19-17-43(3)18-20-44)30-14-11-27(12-15-30)26-9-7-25(8-10-26)24-46-33-6-4-5-32(33)42-36(45)31-21-29(23-41-35(31)39)28-13-16-34(38)40-22-28/h7-16,21-23,32-33H,4-6,17-20,24H2,1-3H3,(H2,39,41)(H,42,45)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298820 (US10125118, Example 226 | US10947215, Example 226) Show SMILES C[C@H](N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C37H43FN6O3/c1-25(44-17-15-43(16-18-44)19-20-45)27-9-11-29(12-10-27)28-7-5-26(6-8-28)24-47-34-4-2-3-33(34)42-37(46)32-21-31(23-41-36(32)39)30-13-14-35(38)40-22-30/h5-14,21-23,25,33-34,45H,2-4,15-20,24H2,1H3,(H2,39,41)(H,42,46)/t25-,33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298821 (US10125118, Example 227 | US10947215, Example 227) Show SMILES C[C@@H](N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C37H43FN6O3/c1-25(44-17-15-43(16-18-44)19-20-45)27-9-11-29(12-10-27)28-7-5-26(6-8-28)24-47-34-4-2-3-33(34)42-37(46)32-21-31(23-41-36(32)39)30-13-14-35(38)40-22-30/h5-14,21-23,25,33-34,45H,2-4,15-20,24H2,1H3,(H2,39,41)(H,42,46)/t25-,33+,34+/m1/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298822 (US10125118, Example 228 | US10947215, Example 228) Show SMILES Nc1ncc(cc1C(=O)N[C@H]1CCC[C@@H]1OCc1ccc(cc1)-c1ccc(cc1)C1(CC1)N1CCN(CCO)CC1)-c1ccc(F)nc1 |r| Show InChI InChI=1S/C38H43FN6O3/c39-35-13-10-29(23-41-35)30-22-32(36(40)42-24-30)37(47)43-33-2-1-3-34(33)48-25-26-4-6-27(7-5-26)28-8-11-31(12-9-28)38(14-15-38)45-18-16-44(17-19-45)20-21-46/h4-13,22-24,33-34,46H,1-3,14-21,25H2,(H2,40,42)(H,43,47)/t33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298823 (US10125118, Example 229 | US10947215, Example 229) Show SMILES CC(C)(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C38H45FN6O3/c1-38(2,45-18-16-44(17-19-45)20-21-46)31-13-10-28(11-14-31)27-8-6-26(7-9-27)25-48-34-5-3-4-33(34)43-37(47)32-22-30(24-42-36(32)40)29-12-15-35(39)41-23-29/h6-15,22-24,33-34,46H,3-5,16-21,25H2,1-2H3,(H2,40,42)(H,43,47)/t33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298824 (US10125118, Example 230 | US10947215, Example 230) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2cncc(F)c2)cc1 |r| Show InChI InChI=1S/C36H41FN6O2/c1-24(43-16-14-42(2)15-17-43)26-10-12-28(13-11-26)27-8-6-25(7-9-27)23-45-34-5-3-4-33(34)41-36(44)32-19-30(21-40-35(32)38)29-18-31(37)22-39-20-29/h6-13,18-22,24,33-34H,3-5,14-17,23H2,1-2H3,(H2,38,40)(H,41,44)/t24?,33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298825 (US10125118, Example 231 | US10947215, Example 231) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(Cl)cnc2N)cc1 |r| Show InChI InChI=1S/C31H38ClN5O2/c1-21(37-16-14-36(2)15-17-37)23-10-12-25(13-11-23)24-8-6-22(7-9-24)20-39-29-5-3-4-28(29)35-31(38)27-18-26(32)19-34-30(27)33/h6-13,18-19,21,28-29H,3-5,14-17,20H2,1-2H3,(H2,33,34)(H,35,38)/t21?,28-,29-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298826 (US10125118, Example 232 | US10947215, Example 232) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(F)cnc2N)cc1 |r| Show InChI InChI=1S/C31H38FN5O2/c1-21(37-16-14-36(2)15-17-37)23-10-12-25(13-11-23)24-8-6-22(7-9-24)20-39-29-5-3-4-28(29)35-31(38)27-18-26(32)19-34-30(27)33/h6-13,18-19,21,28-29H,3-5,14-17,20H2,1-2H3,(H2,33,34)(H,35,38)/t21?,28-,29-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM486602 (US10947215, Example 233) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)C#N)cc1 |r| Show InChI InChI=1S/C32H38N6O2/c1-22(38-16-14-37(2)15-17-38)25-10-12-27(13-11-25)26-8-6-23(7-9-26)21-40-30-5-3-4-29(30)36-32(39)28-18-24(19-33)20-35-31(28)34/h6-13,18,20,22,29-30H,3-5,14-17,21H2,1-2H3,(H2,34,35)(H,36,39)/t22?,29-,30-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298829 (US10125118, Example 235 | US10947215, Example 235) Show SMILES CC(N1CCN(C)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cccnc2N)cc1 |r| Show InChI InChI=1S/C31H39N5O2/c1-22(36-19-17-35(2)18-20-36)24-12-14-26(15-13-24)25-10-8-23(9-11-25)21-38-29-7-3-6-28(29)34-31(37)27-5-4-16-33-30(27)32/h4-5,8-16,22,28-29H,3,6-7,17-21H2,1-2H3,(H2,32,33)(H,34,37)/t22?,28-,29-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298830 (US10125118, Example 236 | US10947215, Example 236) Show SMILES CC(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2cncc(F)c2)cc1 |r| Show InChI InChI=1S/C37H43FN6O3/c1-25(44-15-13-43(14-16-44)17-18-45)27-9-11-29(12-10-27)28-7-5-26(6-8-28)24-47-35-4-2-3-34(35)42-37(46)33-20-31(22-41-36(33)39)30-19-32(38)23-40-21-30/h5-12,19-23,25,34-35,45H,2-4,13-18,24H2,1H3,(H2,39,41)(H,42,46)/t25?,34-,35-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298831 (US10125118, Example 237 | US10947215, Example 237) Show SMILES CC(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2ccc(F)nc2)cc1 |r| Show InChI InChI=1S/C37H43FN6O3/c1-25(44-17-15-43(16-18-44)19-20-45)27-9-11-29(12-10-27)28-7-5-26(6-8-28)24-47-34-4-2-3-33(34)42-37(46)32-21-31(23-41-36(32)39)30-13-14-35(38)40-22-30/h5-14,21-23,25,33-34,45H,2-4,15-20,24H2,1H3,(H2,39,41)(H,42,46)/t25?,33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298832 (US10125118, Example 238 | US10947215, Example 238) Show SMILES CC(N1CCN(CCO)CC1)c1ccc(cc1)-c1ccc(CO[C@H]2CCC[C@@H]2NC(=O)c2cc(cnc2N)-c2cccnc2F)cc1 |r| Show InChI InChI=1S/C37H43FN6O3/c1-25(44-18-16-43(17-19-44)20-21-45)27-11-13-29(14-12-27)28-9-7-26(8-10-28)24-47-34-6-2-5-33(34)42-37(46)32-22-30(23-41-36(32)39)31-4-3-15-40-35(31)38/h3-4,7-15,22-23,25,33-34,45H,2,5-6,16-21,24H2,1H3,(H2,39,41)(H,42,46)/t25?,33-,34-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair
Tyrosine-protein kinase Mer/receptor UFO (Homo sapiens (Human))	BDBM298833 (US10125118, Example 239 | US10947215, Example 239) Show SMILES CN1CCC(Cc2ccc(cc2)-c2ccc(CO[C@H]3CCC[C@@H]3NC(=O)c3cc(cnc3N)-c3cnn(C)c3)cc2)CC1 |r| Show InChI InChI=1S/C35H42N6O2/c1-40-16-14-25(15-17-40)18-24-6-10-27(11-7-24)28-12-8-26(9-13-28)23-43-33-5-3-4-32(33)39-35(42)31-19-29(20-37-34(31)36)30-21-38-41(2)22-30/h6-13,19-22,25,32-33H,3-5,14-18,23H2,1-2H3,(H2,36,37)(H,39,42)/t32-,33-/m0/s1	PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
Dong-A Socio Holdings Co., Ltd. US Patent					Assay Description For the SAR (structure-activity relationship) and compound screening, LanthaScreen™ TR-FRET (Time-Resolved fluorescence energy transfer) assay was em...				US Patent US10947215 (2021) BindingDB Entry DOI: 10.7270/Q2862KKK
					More data for this Ligand-Target Pair

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