Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237471 (US9393232, 2.46) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237443 (US9393232, 2.16) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.60 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237494 (US9393232, 4.1 | US9393232, 4.1a | US9393232, 4.1b) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237509 (US9393232, 2.10a | US9393232, 2.10b) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237521 (US9393232, 2.22) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 32 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237422 (US9393232, 1.30a | US9393232, 1.30b) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 52 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237428 (US9393232, 2.2 | US9393232, 2.2a | US9393232, 2.2b) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 55 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 2 [1-473] (Homo sapiens (Human)) | BDBM237408 (US9393232, 1.16) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 380 | n/a | n/a | n/a | n/a | 7.5 | n/a |
BeiGene, Ltd. US Patent | Assay Description The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K... | US Patent US9393232 (2016) BindingDB Entry DOI: 10.7270/Q25T3JDK | |||||||||||
More data for this Ligand-Target Pair |