Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 2 (MOUSE) | BDBM50023629 (CHEMBL3341861) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258768 (CHEMBL4078901) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 151 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258771 (CHEMBL4062376) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 265 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258826 (CHEMBL4067016) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 299 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258769 (CHEMBL4096928) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 353 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258727 (CHEMBL4081259) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 405 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258738 (CHEMBL4070648) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 439 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258766 (CHEMBL4077975) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 452 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258740 (CHEMBL4085844) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 459 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258767 (CHEMBL4086756) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 464 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258868 (CHEMBL4073727) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 559 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258739 (CHEMBL4064299) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 619 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258781 (CHEMBL4099590) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 651 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258866 (CHEMBL4097779) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 827 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258726 (CHEMBL4078811) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258772 (CHEMBL4091847) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258782 (CHEMBL4071010) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258802 (CHEMBL4089126) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50258770 (CHEMBL4100542) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute , Research Triangle Park, North Carolina 27709, United States. Curated by ChEMBL | Assay Description Allosteric modulation of CB1 receptor in CD-1 mouse cerebellar membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding after 60 m... | J Med Chem 60: 7410-7424 (2017) Article DOI: 10.1021/acs.jmedchem.7b00707 BindingDB Entry DOI: 10.7270/Q2XK8J0H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (MOUSE) | BDBM50323040 (1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylamin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Milano Curated by ChEMBL | Assay Description Inhibition of mouse brain CB2 receptor | Bioorg Med Chem Lett 20: 4406-11 (2010) Article DOI: 10.1016/j.bmcl.2010.06.050 BindingDB Entry DOI: 10.7270/Q24Q7V5B | |||||||||||
More data for this Ligand-Target Pair |