Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q,K548C] (Rattus norvegicus (Rat)) | BDBM214800 (N-methylscopolamine (NMS)) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | 0.555 | n/a | n/a | n/a | 7.4 | n/a |
National Institutes of Health | Assay Description In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing... | J Biol Chem 288: 34777-90 (2013) Article DOI: 10.1074/jbc.M113.503714 BindingDB Entry DOI: 10.7270/Q2JH3K1C | |||||||||||
More data for this Ligand-Target Pair |