Found 96 hits Enz. Inhib. hit(s) with all data for entry = 10841 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573147
![PNG](/data/jpeg/tenK57/BindingDB_573147.png) (US11453673, Example 9)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(CC1)C1CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 0.958 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573138
![PNG](/data/jpeg/tenK57/BindingDB_573138.png) (US11453673, Example 4) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid UniChem
| US Patent
| n/a | n/a | 1.06 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573155
![PNG](/data/jpeg/tenK57/BindingDB_573155.png) (US11453673, Example 16) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573136
![PNG](/data/jpeg/tenK57/BindingDB_573136.png) (US11453673, Example 3) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 1.26 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573154
![PNG](/data/jpeg/tenK57/BindingDB_573154.png) (US11453673, Example 15)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1(C)CC1)C1(CC1)C1CC1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573144
![PNG](/data/jpeg/tenK57/BindingDB_573144.png) (US11453673, Example 6)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1CCCCO1)C1(CC1)C1CC1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 1.88 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573148
![PNG](/data/jpeg/tenK57/BindingDB_573148.png) (US11453673, Example 10)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(CC1)C1CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573139
![PNG](/data/jpeg/tenK57/BindingDB_573139.png) (US11453673, Example 5) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573135
![PNG](/data/jpeg/tenK57/BindingDB_573135.png) (US11453673, Example 2) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 2.81 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573154
![PNG](/data/jpeg/tenK57/BindingDB_573154.png) (US11453673, Example 15)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1(C)CC1)C1(CC1)C1CC1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573138
![PNG](/data/jpeg/tenK57/BindingDB_573138.png) (US11453673, Example 4) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid UniChem
| US Patent
| n/a | n/a | 3.65 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573138
![PNG](/data/jpeg/tenK57/BindingDB_573138.png) (US11453673, Example 4) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid UniChem
| US Patent
| n/a | n/a | 3.71 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573135
![PNG](/data/jpeg/tenK57/BindingDB_573135.png) (US11453673, Example 2) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 3.73 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573147
![PNG](/data/jpeg/tenK57/BindingDB_573147.png) (US11453673, Example 9)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(CC1)C1CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 3.73 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573135
![PNG](/data/jpeg/tenK57/BindingDB_573135.png) (US11453673, Example 2) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 4.11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573149
![PNG](/data/jpeg/tenK57/BindingDB_573149.png) (US11453673, Example 11)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@@H]1CCCCO1)c2=O |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 4.77 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573154
![PNG](/data/jpeg/tenK57/BindingDB_573154.png) (US11453673, Example 15)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1(C)CC1)C1(CC1)C1CC1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573147
![PNG](/data/jpeg/tenK57/BindingDB_573147.png) (US11453673, Example 9)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(CC1)C1CC1 |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 4.94 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573144
![PNG](/data/jpeg/tenK57/BindingDB_573144.png) (US11453673, Example 6)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1CCCCO1)C1(CC1)C1CC1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 5.98 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573152
![PNG](/data/jpeg/tenK57/BindingDB_573152.png) (US11453673, Example 13)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(C)CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 6.35 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573155
![PNG](/data/jpeg/tenK57/BindingDB_573155.png) (US11453673, Example 16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 6.54 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573148
![PNG](/data/jpeg/tenK57/BindingDB_573148.png) (US11453673, Example 10)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(CC1)C1CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 6.72 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573144
![PNG](/data/jpeg/tenK57/BindingDB_573144.png) (US11453673, Example 6)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1CC1CCCCO1)C1(CC1)C1CC1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 7.03 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573145
![PNG](/data/jpeg/tenK57/BindingDB_573145.png) (US11453673, Example 7) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 7.76 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573155
![PNG](/data/jpeg/tenK57/BindingDB_573155.png) (US11453673, Example 16) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 8.67 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573136
![PNG](/data/jpeg/tenK57/BindingDB_573136.png) (US11453673, Example 3) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 9.36 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573146
![PNG](/data/jpeg/tenK57/BindingDB_573146.png) (US11453673, Example 8) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 10.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573148
![PNG](/data/jpeg/tenK57/BindingDB_573148.png) (US11453673, Example 10)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(CC1)C1CC1 |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573136
![PNG](/data/jpeg/tenK57/BindingDB_573136.png) (US11453673, Example 3) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573139
![PNG](/data/jpeg/tenK57/BindingDB_573139.png) (US11453673, Example 5) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 11.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573139
![PNG](/data/jpeg/tenK57/BindingDB_573139.png) (US11453673, Example 5) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573134
![PNG](/data/jpeg/tenK57/BindingDB_573134.png) (US11453673, Example 1)Show SMILES Cn1cc(Cc2cn3c(nnc3c(=O)n2CC2CC2)C2(CC2)C2CC2)cn1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573149
![PNG](/data/jpeg/tenK57/BindingDB_573149.png) (US11453673, Example 11)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@@H]1CCCCO1)c2=O |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 13.2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573150
![PNG](/data/jpeg/tenK57/BindingDB_573150.png) (US11453673, Example 12)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@H]1CCCCO1)c2=O |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 13.2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573149
![PNG](/data/jpeg/tenK57/BindingDB_573149.png) (US11453673, Example 11)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@@H]1CCCCO1)c2=O |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 17.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573134
![PNG](/data/jpeg/tenK57/BindingDB_573134.png) (US11453673, Example 1)Show SMILES Cn1cc(Cc2cn3c(nnc3c(=O)n2CC2CC2)C2(CC2)C2CC2)cn1 | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 20.3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573152
![PNG](/data/jpeg/tenK57/BindingDB_573152.png) (US11453673, Example 13)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(C)CC1 |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 21.8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573152
![PNG](/data/jpeg/tenK57/BindingDB_573152.png) (US11453673, Example 13)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@@H]1CCCCO1)C1(C)CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 21.8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C
(Homo sapiens (Human)) | BDBM573153
![PNG](/data/jpeg/tenK57/BindingDB_573153.png) (US11453673, Example 14)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(C)CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 22.3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573146
![PNG](/data/jpeg/tenK57/BindingDB_573146.png) (US11453673, Example 8) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 25.4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573145
![PNG](/data/jpeg/tenK57/BindingDB_573145.png) (US11453673, Example 7) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 28.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573134
![PNG](/data/jpeg/tenK57/BindingDB_573134.png) (US11453673, Example 1)Show SMILES Cn1cc(Cc2cn3c(nnc3c(=O)n2CC2CC2)C2(CC2)C2CC2)cn1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 29.4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573145
![PNG](/data/jpeg/tenK57/BindingDB_573145.png) (US11453673, Example 7) | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 32.7 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573150
![PNG](/data/jpeg/tenK57/BindingDB_573150.png) (US11453673, Example 12)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@H]1CCCCO1)c2=O |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 33.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573146
![PNG](/data/jpeg/tenK57/BindingDB_573146.png) (US11453673, Example 8) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 36.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573150
![PNG](/data/jpeg/tenK57/BindingDB_573150.png) (US11453673, Example 12)Show SMILES CCC1(CC1)c1nnc2n1c(C)c(C)n(C[C@H]1CCCCO1)c2=O |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 44.6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
(Homo sapiens (Human)) | BDBM573153
![PNG](/data/jpeg/tenK57/BindingDB_573153.png) (US11453673, Example 14)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(C)CC1 |r| | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
(Homo sapiens (Human)) | BDBM573153
![PNG](/data/jpeg/tenK57/BindingDB_573153.png) (US11453673, Example 14)Show SMILES Cc1c(C)n2c(nnc2c(=O)n1C[C@H]1CCCCO1)C1(C)CC1 |r| | KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 52.4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description TABLE 5: All 3′, 5′ cyclic nucleotide PDE enzyme activities are measured with a radiometric enzyme assay based on SPA detection system. C... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha/beta
(Homo sapiens (Human)) | BDBM573146
![PNG](/data/jpeg/tenK57/BindingDB_573146.png) (US11453673, Example 8) | PDB
UniProtKB/SwissProt
antibodypedia antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 2.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Table 7: The following phosphodiesterase activities are measured using [3H]cGMP as reaction substrate: human PDE6A/6B. The catalytic active form of h... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4D
(Homo sapiens (Human)) | BDBM573134
![PNG](/data/jpeg/tenK57/BindingDB_573134.png) (US11453673, Example 1)Show SMILES Cn1cc(Cc2cn3c(nnc3c(=O)n2CC2CC2)C2(CC2)C2CC2)cn1 | PDB
KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| US Patent
| n/a | n/a | 5.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Table 6: The following PDE activities are measured using [3H]cAMP as reaction substrate: human PDE3A (catalytic domain) and human PDE4D. Both enzymes... |
Citation and Details
BindingDB Entry DOI: 10.7270/Q22Z18RF |
More data for this Ligand-Target Pair | |