BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 124 hits Enz. Inhib. hit(s) with all data for entry = 1428   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322581
PNG
(US10183940, Example 33)
Show SMILES Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-13-6-4-8-15-17(13)24-25-19(15)21(2,3)23-20(26)16-9-5-7-14-12-22-10-11-27-18(14)16/h4-9,22H,10-12H2,1-3H3,(H,23,26)(H,24,25)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
21.7n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322587
PNG
(US10183940, Example 39)
Show SMILES Cn1nc(c2cccc(F)c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H23FN4O2/c1-21(2,19-14-7-5-9-16(22)17(14)26(3)25-19)24-20(27)15-8-4-6-13-12-23-10-11-28-18(13)15/h4-9,23H,10-12H2,1-3H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
29.1n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322565
PNG
(US10183940, Example 18)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-21(2,19-15-8-4-5-10-17(15)25(3)24-19)23-20(26)16-9-6-7-14-13-22-11-12-27-18(14)16/h4-10,22H,11-13H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
39.5n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
53.2n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322573
PNG
(US10183940, Example 26)
Show SMILES Cc1nnc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-16-8-4-5-9-17(16)20(26-25-14)22(2,3)24-21(27)18-10-6-7-15-13-23-11-12-28-19(15)18/h4-10,23H,11-13H2,1-3H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
65n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322553
PNG
(US10183940, Example 6)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ccnc2ccccc12
Show InChI InChI=1S/C22H23N3O2/c1-22(2,18-10-11-24-19-9-4-3-7-16(18)19)25-21(26)17-8-5-6-15-14-23-12-13-27-20(15)17/h3-11,23H,12-14H2,1-2H3,(H,25,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
104n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322590
PNG
(US10183940, Example 42)
Show SMILES Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)c1cncc2CNCCOc12
Show InChI InChI=1S/C21H25N5O2/c1-13-6-5-7-15-17(13)26(4)25-19(15)21(2,3)24-20(27)16-12-23-11-14-10-22-8-9-28-18(14)16/h5-7,11-12,22H,8-10H2,1-4H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
532n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322567
PNG
(US10183940, Example 20)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1ccnc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-13-6-4-5-7-16(13)25(3)24-18)23-19(26)14-8-9-22-15-12-21-10-11-27-17(14)15/h4-9,21H,10-12H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
574n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322566
PNG
(US10183940, Example 19)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1nccc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-14-6-4-5-7-15(14)25(3)24-18)23-19(26)16-17-13(8-9-22-16)12-21-10-11-27-17/h4-9,21H,10-12H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
613n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322565
PNG
(US10183940, Example 18)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-21(2,19-15-8-4-5-10-17(15)25(3)24-19)23-20(26)16-9-6-7-14-13-22-11-12-27-18(14)16/h4-10,22H,11-13H2,1-3H3,(H,23,26)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
7.82E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322567
PNG
(US10183940, Example 20)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1ccnc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-13-6-4-5-7-16(13)25(3)24-18)23-19(26)14-8-9-22-15-12-21-10-11-27-17(14)15/h4-9,21H,10-12H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.62E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322566
PNG
(US10183940, Example 19)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1nccc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-14-6-4-5-7-15(14)25(3)24-18)23-19(26)16-17-13(8-9-22-16)12-21-10-11-27-17/h4-9,21H,10-12H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.62E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322581
PNG
(US10183940, Example 33)
Show SMILES Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-13-6-4-8-15-17(13)24-25-19(15)21(2,3)23-20(26)16-9-5-7-14-12-22-10-11-27-18(14)16/h4-9,22H,10-12H2,1-3H3,(H,23,26)(H,24,25)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.62E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322573
PNG
(US10183940, Example 26)
Show SMILES Cc1nnc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-16-8-4-5-9-17(16)20(26-25-14)22(2,3)24-21(27)18-10-6-7-15-13-23-11-12-28-19(15)18/h4-10,23H,11-13H2,1-3H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.62E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322590
PNG
(US10183940, Example 42)
Show SMILES Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)c1cncc2CNCCOc12
Show InChI InChI=1S/C21H25N5O2/c1-13-6-5-7-15-17(13)26(4)25-19(15)21(2,3)24-20(27)16-12-23-11-14-10-22-8-9-28-18(14)16/h5-7,11-12,22H,8-10H2,1-4H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.62E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322553
PNG
(US10183940, Example 6)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ccnc2ccccc12
Show InChI InChI=1S/C22H23N3O2/c1-22(2,18-10-11-24-19-9-4-3-7-16(18)19)25-21(26)17-8-5-6-15-14-23-12-13-27-20(15)17/h3-11,23H,12-14H2,1-2H3,(H,25,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.71E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.71E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322565
PNG
(US10183940, Example 18)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-21(2,19-15-8-4-5-10-17(15)25(3)24-19)23-20(26)16-9-6-7-14-13-22-11-12-27-18(14)16/h4-10,22H,11-13H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.71E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 3


(Homo sapiens (Human))
BDBM322587
PNG
(US10183940, Example 39)
Show SMILES Cn1nc(c2cccc(F)c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H23FN4O2/c1-21(2,19-14-7-5-9-16(22)17(14)26(3)25-19)24-20(27)15-8-4-6-13-12-23-10-11-28-18(13)15/h4-9,23H,10-12H2,1-3H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
8.71E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322553
PNG
(US10183940, Example 6)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ccnc2ccccc12
Show InChI InChI=1S/C22H23N3O2/c1-22(2,18-10-11-24-19-9-4-3-7-16(18)19)25-21(26)17-8-5-6-15-14-23-12-13-27-20(15)17/h3-11,23H,12-14H2,1-2H3,(H,25,26)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.01E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.01E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322587
PNG
(US10183940, Example 39)
Show SMILES Cn1nc(c2cccc(F)c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H23FN4O2/c1-21(2,19-14-7-5-9-16(22)17(14)26(3)25-19)24-20(27)15-8-4-6-13-12-23-10-11-28-18(13)15/h4-9,23H,10-12H2,1-3H3,(H,24,27)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.01E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322567
PNG
(US10183940, Example 20)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1ccnc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-13-6-4-5-7-16(13)25(3)24-18)23-19(26)14-8-9-22-15-12-21-10-11-27-17(14)15/h4-9,21H,10-12H2,1-3H3,(H,23,26)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.45E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322573
PNG
(US10183940, Example 26)
Show SMILES Cc1nnc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-16-8-4-5-9-17(16)20(26-25-14)22(2,3)24-21(27)18-10-6-7-15-13-23-11-12-28-19(15)18/h4-10,23H,11-13H2,1-3H3,(H,24,27)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.45E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322566
PNG
(US10183940, Example 19)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1nccc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-14-6-4-5-7-15(14)25(3)24-18)23-19(26)16-17-13(8-9-22-16)12-21-10-11-27-17/h4-9,21H,10-12H2,1-3H3,(H,23,26)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.45E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322581
PNG
(US10183940, Example 33)
Show SMILES Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-13-6-4-8-15-17(13)24-25-19(15)21(2,3)23-20(26)16-9-5-7-14-12-22-10-11-27-18(14)16/h4-9,22H,10-12H2,1-3H3,(H,23,26)(H,24,25)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.45E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 1


(Homo sapiens (Human))
BDBM322590
PNG
(US10183940, Example 42)
Show SMILES Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)c1cncc2CNCCOc12
Show InChI InChI=1S/C21H25N5O2/c1-13-6-5-7-15-17(13)26(4)25-19(15)21(2,3)24-20(27)16-12-23-11-14-10-22-8-9-28-18(14)16/h5-7,11-12,22H,8-10H2,1-4H3,(H,24,27)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.45E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322566
PNG
(US10183940, Example 19)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1nccc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-14-6-4-5-7-15(14)25(3)24-18)23-19(26)16-17-13(8-9-22-16)12-21-10-11-27-17/h4-9,21H,10-12H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.60E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322590
PNG
(US10183940, Example 42)
Show SMILES Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)c1cncc2CNCCOc12
Show InChI InChI=1S/C21H25N5O2/c1-13-6-5-7-15-17(13)26(4)25-19(15)21(2,3)24-20(27)16-12-23-11-14-10-22-8-9-28-18(14)16/h5-7,11-12,22H,8-10H2,1-4H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.60E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322581
PNG
(US10183940, Example 33)
Show SMILES Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-13-6-4-8-15-17(13)24-25-19(15)21(2,3)23-20(26)16-9-5-7-14-12-22-10-11-27-18(14)16/h4-9,22H,10-12H2,1-3H3,(H,23,26)(H,24,25)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.60E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322573
PNG
(US10183940, Example 26)
Show SMILES Cc1nnc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-16-8-4-5-9-17(16)20(26-25-14)22(2,3)24-21(27)18-10-6-7-15-13-23-11-12-28-19(15)18/h4-10,23H,11-13H2,1-3H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.60E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322567
PNG
(US10183940, Example 20)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1ccnc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-13-6-4-5-7-16(13)25(3)24-18)23-19(26)14-8-9-22-15-12-21-10-11-27-17(14)15/h4-9,21H,10-12H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.60E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.63E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322587
PNG
(US10183940, Example 39)
Show SMILES Cn1nc(c2cccc(F)c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H23FN4O2/c1-21(2,19-14-7-5-9-16(22)17(14)26(3)25-19)24-20(27)15-8-4-6-13-12-23-10-11-28-18(13)15/h4-9,23H,10-12H2,1-3H3,(H,24,27)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.63E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322553
PNG
(US10183940, Example 6)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ccnc2ccccc12
Show InChI InChI=1S/C22H23N3O2/c1-22(2,18-10-11-24-19-9-4-3-7-16(18)19)25-21(26)17-8-5-6-15-14-23-12-13-27-20(15)17/h3-11,23H,12-14H2,1-2H3,(H,25,26)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.63E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 2


(Homo sapiens (Human))
BDBM322565
PNG
(US10183940, Example 18)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-21(2,19-15-8-4-5-10-17(15)25(3)24-19)23-20(26)16-9-6-7-14-13-22-11-12-27-18(14)16/h4-10,22H,11-13H2,1-3H3,(H,23,26)
PDB

KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.63E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322590
PNG
(US10183940, Example 42)
Show SMILES Cc1cccc2c(nn(C)c12)C(C)(C)NC(=O)c1cncc2CNCCOc12
Show InChI InChI=1S/C21H25N5O2/c1-13-6-5-7-15-17(13)26(4)25-19(15)21(2,3)24-20(27)16-12-23-11-14-10-22-8-9-28-18(14)16/h5-7,11-12,22H,8-10H2,1-4H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.75E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322573
PNG
(US10183940, Example 26)
Show SMILES Cc1nnc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-16-8-4-5-9-17(16)20(26-25-14)22(2,3)24-21(27)18-10-6-7-15-13-23-11-12-28-19(15)18/h4-10,23H,11-13H2,1-3H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.75E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322567
PNG
(US10183940, Example 20)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1ccnc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-13-6-4-5-7-16(13)25(3)24-18)23-19(26)14-8-9-22-15-12-21-10-11-27-17(14)15/h4-9,21H,10-12H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.75E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322581
PNG
(US10183940, Example 33)
Show SMILES Cc1cccc2c(n[nH]c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-13-6-4-8-15-17(13)24-25-19(15)21(2,3)23-20(26)16-9-5-7-14-12-22-10-11-27-18(14)16/h4-9,22H,10-12H2,1-3H3,(H,23,26)(H,24,25)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.75E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322566
PNG
(US10183940, Example 19)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1nccc2CNCCOc12
Show InChI InChI=1S/C20H23N5O2/c1-20(2,18-14-6-4-5-7-15(14)25(3)24-18)23-19(26)16-17-13(8-9-22-16)12-21-10-11-27-17/h4-9,21H,10-12H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.75E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322565
PNG
(US10183940, Example 18)
Show SMILES Cn1nc(c2ccccc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-21(2,19-15-8-4-5-10-17(15)25(3)24-19)23-20(26)16-9-6-7-14-13-22-11-12-27-18(14)16/h4-10,22H,11-13H2,1-3H3,(H,23,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.86E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322587
PNG
(US10183940, Example 39)
Show SMILES Cn1nc(c2cccc(F)c12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H23FN4O2/c1-21(2,19-14-7-5-9-16(22)17(14)26(3)25-19)24-20(27)15-8-4-6-13-12-23-10-11-28-18(13)15/h4-9,23H,10-12H2,1-3H3,(H,24,27)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.86E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.86E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 5


(Homo sapiens (Human))
BDBM322553
PNG
(US10183940, Example 6)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ccnc2ccccc12
Show InChI InChI=1S/C22H23N3O2/c1-22(2,18-10-11-24-19-9-4-3-7-16(18)19)25-21(26)17-8-5-6-15-14-23-12-13-27-20(15)17/h3-11,23H,12-14H2,1-2H3,(H,25,26)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
9.86E+3n/an/an/an/an/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
Method description for binding assays with human Somatostatin receptors by use of CHO cell membranes expressing recombinant human SSTR1 or human SSTR...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322592
PNG
(US10183940, Example 44)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1n[nH]c2c(Cl)cccc12
Show InChI InChI=1S/C20H21ClN4O2/c1-20(2,18-13-6-4-8-15(21)16(13)24-25-18)23-19(26)14-7-3-5-12-11-22-9-10-27-17(12)14/h3-8,22H,9-11H2,1-2H3,(H,23,26)(H,24,25)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 1.30n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322593
PNG
(US10183940, Example 45)
Show SMILES Cc1cccc2c(ncnc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C22H24N4O2/c1-14-6-4-8-16-18(14)24-13-25-20(16)22(2,3)26-21(27)17-9-5-7-15-12-23-10-11-28-19(15)17/h4-9,13,23H,10-12H2,1-3H3,(H,26,27)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 9.20n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322594
PNG
(US10183940, Example 46)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ncnc2ccccc12
Show InChI InChI=1S/C21H22N4O2/c1-21(2,19-15-7-3-4-9-17(15)23-13-24-19)25-20(26)16-8-5-6-14-12-22-10-11-27-18(14)16/h3-9,13,22H,10-12H2,1-2H3,(H,25,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 9.20n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322595
PNG
(US10183940, Example 47)
Show SMILES Cc1cccn2c(ncc12)C(C)(C)NC(=O)c1cccc2CNCCOc12
Show InChI InChI=1S/C21H24N4O2/c1-14-6-5-10-25-17(14)13-23-20(25)21(2,3)24-19(26)16-8-4-7-15-12-22-9-11-27-18(15)16/h4-8,10,13,22H,9,11-12H2,1-3H3,(H,24,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 2n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Somatostatin receptor type 4


(Homo sapiens (Human))
BDBM322596
PNG
(US10183940, Example 48)
Show SMILES CC(C)(NC(=O)c1cccc2CNCCOc12)c1ncc2c(Cl)cccn12
Show InChI InChI=1S/C20H21ClN4O2/c1-20(2,19-23-12-16-15(21)7-4-9-25(16)19)24-18(26)14-6-3-5-13-11-22-8-10-27-17(13)14/h3-7,9,12,22H,8,10-11H2,1-2H3,(H,24,26)
PDB

KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 1.70n/an/an/an/a



Boehringer Ingelheim International GmbH

US Patent


Assay Description
The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...


US Patent US10183940 (2019)


BindingDB Entry DOI: 10.7270/Q2KW5J45
More data for this
Ligand-Target Pair
Displayed 1 to 50 (of 124 total )  |  Next  |  Last  >>
Jump to: