Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520104 (CHEMBL4535971) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Inhibition of human EP4 transfected in human HEK293 cells co transfected with SmBit-beta-arrestin. assessed as reduction in PGE2 induced-beta-arresti... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520069 (CHEMBL4457944) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520101 (CHEMBL4439228) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520098 (CHEMBL4548291) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520104 (CHEMBL4535971) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Inhibition of human EP4 transfected in human HEK293 cells co transfected with CRE-luciferase assessed as reduction in PGE2-induced luciferase express... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520104 (CHEMBL4535971) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM119448 (US8686018, 107) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.5 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520086 (CHEMBL4463343) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520114 (CHEMBL4462095) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520103 (CHEMBL4455965) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520097 (CHEMBL4564092) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520072 (CHEMBL4550862) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520100 (CHEMBL4576681) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520104 (CHEMBL4535971) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520104 (CHEMBL4535971) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Inhibition of human EP4 transfected in human HEK293 cells assessed as reduction in PGE2-induced cAMP level incubated for 15 mins followed by PGE2 sti... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520110 (CHEMBL4569593) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520097 (CHEMBL4564092) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520102 (CHEMBL4453648) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520090 (CHEMBL4442135) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520073 (CHEMBL4591792) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520100 (CHEMBL4576681) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520098 (CHEMBL4548291) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520071 (CHEMBL4440382) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520091 (CHEMBL4574900) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520112 (CHEMBL4519666) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520071 (CHEMBL4440382) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520070 (CHEMBL4568156) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520119 (CHEMBL4466382) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520109 (CHEMBL4562090) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520073 (CHEMBL4591792) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520094 (CHEMBL4589657) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520089 (CHEMBL4455816) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520096 (CHEMBL4553892) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 119 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520111 (CHEMBL4544033) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 119 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520103 (CHEMBL4455965) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520101 (CHEMBL4439228) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520069 (CHEMBL4457944) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 135 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520088 (CHEMBL4448318) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 148 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520095 (CHEMBL4545487) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 161 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM119448 (US8686018, 107) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 181 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520118 (CHEMBL4573602) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 183 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520072 (CHEMBL4550862) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520082 (CHEMBL4450391) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 225 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520108 (CHEMBL4468734) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 276 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520087 (CHEMBL4443888) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520102 (CHEMBL4453648) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520115 (CHEMBL4442888) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 647 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Mus musculus (Mouse)) | BDBM50520086 (CHEMBL4463343) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 906 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520113 (CHEMBL4440611) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP4 subtype (Homo sapiens (Human)) | BDBM50520099 (CHEMBL4563586) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
East China Normal University Curated by ChEMBL | Assay Description Antagonist activity at human EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow... | J Med Chem 63: 569-590 (2020) Article DOI: 10.1021/acs.jmedchem.9b01269 BindingDB Entry DOI: 10.7270/Q2N58QRT | |||||||||||
More data for this Ligand-Target Pair |
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