Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583918 (CHEMBL4791134) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583916 (CHEMBL4786320) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50526790 (CHEMBL4555799) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583916 (CHEMBL4786320) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50526790 (CHEMBL4555799) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583918 (CHEMBL4791134) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583925 (CHEMBL4782954) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583922 (CHEMBL4786555) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583922 (CHEMBL4786555) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583916 (CHEMBL4786320) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583922 (CHEMBL4786555) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583925 (CHEMBL4782954) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583919 (CHEMBL5083688) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583921 (CHEMBL4779443) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583920 (CHEMBL4786843) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583927 (CHEMBL5088381) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583918 (CHEMBL4791134) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 78 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583919 (CHEMBL5083688) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583927 (CHEMBL5088381) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583920 (CHEMBL4786843) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 95 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50526790 (CHEMBL4555799) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583923 (CHEMBL4786592) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583924 (CHEMBL4790490) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 112 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583920 (CHEMBL4786843) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 128 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583921 (CHEMBL4779443) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 133 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583917 (CHEMBL4800180) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 135 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583924 (CHEMBL4790490) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 138 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583928 (CHEMBL5080711) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 156 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583927 (CHEMBL5088381) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 189 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583926 (CHEMBL4798916) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 215 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583925 (CHEMBL4782954) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 284 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583923 (CHEMBL4786592) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 286 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583921 (CHEMBL4779443) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 299 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583919 (CHEMBL5083688) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 347 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583923 (CHEMBL4786592) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 414 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583917 (CHEMBL4800180) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583924 (CHEMBL4790490) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583928 (CHEMBL5080711) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 572 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583928 (CHEMBL5080711) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 771 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583926 (CHEMBL4798916) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 907 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583917 (CHEMBL4800180) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 923 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583926 (CHEMBL4798916) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 12 (Homo sapiens) | BDBM50583929 (SY-5609 | SY5609 | Sy 5609 | Sy-5609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50583929 (SY-5609 | SY5609 | Sy 5609 | Sy-5609) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Homo sapiens (Human)) | BDBM50583929 (SY-5609 | SY5609 | Sy 5609 | Sy-5609) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 5.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assay | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-H/Cyclin-dependent kinase 7 (Homo sapiens (Human)) | BDBM50526790 (CHEMBL4555799) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.330 | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Binding affinity to full length CDK7 (1 to 346 residues) /N-terminal TEV cleavable 6His tagged full length cyclinH (1 to 323 residues) (unknown origi... | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-H/Cyclin-dependent kinase 7 (Homo sapiens (Human)) | BDBM50583919 (CHEMBL5083688) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Binding affinity to full length CDK7 (1 to 346 residues) /N-terminal TEV cleavable 6His tagged full length cyclinH (1 to 323 residues) (unknown origi... | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-H/Cyclin-dependent kinase 7 (Homo sapiens (Human)) | BDBM50583920 (CHEMBL4786843) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.340 | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Binding affinity to full length CDK7 (1 to 346 residues) /N-terminal TEV cleavable 6His tagged full length cyclinH (1 to 323 residues) (unknown origi... | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-H/Cyclin-dependent kinase 7 (Homo sapiens (Human)) | BDBM50583921 (CHEMBL4779443) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Binding affinity to full length CDK7 (1 to 346 residues) /N-terminal TEV cleavable 6His tagged full length cyclinH (1 to 323 residues) (unknown origi... | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-H/Cyclin-dependent kinase 7 (Homo sapiens (Human)) | BDBM50583917 (CHEMBL4800180) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a |
Institute of Medicinal Molecular Design, Inc. Curated by ChEMBL | Assay Description Binding affinity to full length CDK7 (1 to 346 residues) /N-terminal TEV cleavable 6His tagged full length cyclinH (1 to 323 residues) (unknown origi... | J Med Chem 47: 4818-28 (2004) Article DOI: 10.1021/acs.jmedchem.1c01171 BindingDB Entry DOI: 10.7270/Q2736VSR | |||||||||||
More data for this Ligand-Target Pair |
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