Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Corticotropin-releasing factor receptor 2 (Mus musculus) | BDBM50075918 (8N-[2-amino-(1R,2R)-cyclohexyl]-15-oxo-(9aS,13aS)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 86 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
A Subsidiary of Agouron Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 beta | Bioorg Med Chem Lett 9: 765-70 (1999) BindingDB Entry DOI: 10.7270/Q2TD9WJJ | |||||||||||
More data for this Ligand-Target Pair |