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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Ghrelin O-acyltransferase' and Ligand = 'BDBM50548079'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Ghrelin O-acyltransferase


(Homo sapiens (Human))		BDBM50548079
PNG
(CHEMBL4754865)
Show SMILES COc1cc(ccc1Cc1c(C)nc2nonc2c1N)C(F)(F)F
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 0.0660n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISA

Citation and Details

Article DOI: 10.1039/d0md00210k
BindingDB Entry DOI: 10.7270/Q2KS6W53
More data for this
Ligand-Target Pair