BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Importin subunit alpha-1' and Ligand = 'BDBM75033'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Importin subunit alpha-1


(Homo sapiens (Human))
BDBM75033
PNG
(5-({[(1-methyl-1H-tetrazol-5-yl)thio]acetyl}amino)...)
Show SMILES Cn1nnnc1SCC(=O)Nc1nn(nc1C(N)=O)-c1ccccc1
Show InChI InChI=1S/C13H13N9O2S/c1-21-13(16-19-20-21)25-7-9(23)15-12-10(11(14)24)17-22(18-12)8-5-3-2-4-6-8/h2-6H,7H2,1H3,(H2,14,24)(H,15,18,23)
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
PCBioAssay
n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...


PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair