Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Isoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E] (Homo sapiens (Human)) | BDBM65501![]() (8-pCP-cGMP | Cyclic GMP analogs | cGMP) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 7.70 | n/a | n/a | 7.0 | n/a |
Baylor College of Medicine | Assay Description Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ... | ACS Chem Biol 12: 2388-2398 (2017) Article DOI: 10.1021/acschembio.7b00369 BindingDB Entry DOI: 10.7270/Q2930RB1 | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Isoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E] (Homo sapiens (Human)) | BDBM65501![]() (8-pCP-cGMP | Cyclic GMP analogs | cGMP) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 4.20 | n/a | n/a | 7.0 | n/a |
Baylor College of Medicine | Assay Description Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ... | ACS Chem Biol 12: 2388-2398 (2017) Article DOI: 10.1021/acschembio.7b00369 BindingDB Entry DOI: 10.7270/Q2930RB1 | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |