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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM301791'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mast/stem cell growth factor receptor Kit


(Homo sapiens (Human))		BDBM301791
PNG
(N-[6-(2-Benzyloxy-ethoxy)-1H-indazol-3-yl]-(1-meth...)
Show SMILES CN1CCC(CC1)Nc1ccccc1C(=O)Nc1n[nH]c2cc(OCCOCc3ccccc3)ccc12
Show InChI InChI=1S/C29H33N5O3/c1-34-15-13-22(14-16-34)30-26-10-6-5-9-25(26)29(35)31-28-24-12-11-23(19-27(24)32-33-28)37-18-17-36-20-21-7-3-2-4-8-21/h2-12,19,22,30H,13-18,20H2,1H3,(H2,31,32,33,35)
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 61n/an/an/an/an/an/a



NERVIANO MEDICAL SCIENCES S.R.L.

US Patent


Assay Description
i. Enzyme The assay has been performed using KIT cytoplasmic domain product and purified in house as GST fused protein. The KIT protein (4.5 microM) ...

US Patent US9597317 (2017)


BindingDB Entry DOI: 10.7270/Q2N58PDX
More data for this
Ligand-Target Pair