Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM392409'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Mast/stem cell growth factor receptor Kit (Homo sapiens (Human))	BDBM392409 (3-methyl-N-(2-morpholino-1H- pyrrolo[2,3-b]pyridin...) Show SMILES Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)N1CCOCC1 Show InChI InChI=1S/C16H18N6O2/c1-10-6-13(21-20-10)16(23)18-12-7-11-8-14(19-15(11)17-9-12)22-2-4-24-5-3-22/h6-9H,2-5H2,1H3,(H,17,19)(H,18,23)(H,20,21)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	<1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...				J Med Chem 52: 1799-802 (2009) BindingDB Entry DOI: 10.7270/Q2HH6NDZ
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