Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412177 (CHEMBL493979) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412177 (CHEMBL493979) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair |