Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50105697![]() (1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human platelets | Bioorg Med Chem Lett 11: 2851-3 (2001) BindingDB Entry DOI: 10.7270/Q2NP23PC | |||||||||||
More data for this Ligand-Target Pair |