Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase K103N mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complex | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase L100I mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complex | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 free reverse transcriptase L100I mutant | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase L100I mutant/poly(rA)/oligo(dT) DNA binary complex | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase K103N mutant/poly(rA)/oligo(dT) DNA binary complex | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 free reverse transcriptase K103N mutant | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase K103N mutant | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase protein (Human immunodeficiency virus 1) | BDBM50339536 ((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
2-Universit£ di Siena Curated by ChEMBL | Assay Description Inhibition of HIV1 reverse transcriptase L100I mutant | Bioorg Med Chem Lett 21: 3935-8 (2011) Article DOI: 10.1016/j.bmcl.2011.05.020 BindingDB Entry DOI: 10.7270/Q2319ZQ9 | |||||||||||
More data for this Ligand-Target Pair |