Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase PLK3 (Homo sapiens (Human)) | BDBM50519158 (CHEMBL4445812) | PDB NCI pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 456 | n/a | n/a | n/a | n/a | n/a |
Chengdu University Curated by ChEMBL | Assay Description Binding affinity to wild-type human partial length PLK3 (A42 to L334 residues) expressed in mammalian expression system measured after 1 hr by kinome... | J Med Chem 62: 7697-7707 (2019) Article DOI: 10.1021/acs.jmedchem.9b00353 BindingDB Entry DOI: 10.7270/Q2X06BF7 | |||||||||||
More data for this Ligand-Target Pair |