Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50046751 (CHEMBL3309646) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CSIR-Indian Institute of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of bovine brain tubulin polymerization measured for 1 hr at 1 min intervals by fluorescence assay | Bioorg Med Chem Lett 24: 3356-60 (2014) Article DOI: 10.1016/j.bmcl.2014.05.096 BindingDB Entry DOI: 10.7270/Q2X068PJ | |||||||||||
More data for this Ligand-Target Pair |