Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcriptional enhancer factor TEF-3 (Homo sapiens) | BDBM50535724 (CHEMBL4467555) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Inhibition of human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) interaction with N-biotinylated YAP (60 to 100 residues) inc... | Bioorg Med Chem Lett 29: 2316-2319 (2019) Article DOI: 10.1016/j.bmcl.2019.06.022 BindingDB Entry DOI: 10.7270/Q2WH2TH8 | |||||||||||
More data for this Ligand-Target Pair |