Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transitional endoplasmic reticulum ATPase (Homo sapiens (Human)) | BDBM50500324![]() (CHEMBL3747448) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Curated by ChEMBL | Assay Description Inhibition of His-tagged p97 (unknown origin) in presence of ATP and PNP by UV-transparent microplate assay | J Med Chem 62: 2814-2829 (2019) Article DOI: 10.1021/acs.jmedchem.9b00144 BindingDB Entry DOI: 10.7270/Q24171H0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transitional endoplasmic reticulum ATPase (Homo sapiens (Human)) | BDBM50500324![]() (CHEMBL3747448) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Cleave Biosciences Inc. Curated by ChEMBL | Assay Description Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assay | J Med Chem 58: 9480-97 (2015) Article DOI: 10.1021/acs.jmedchem.5b01346 BindingDB Entry DOI: 10.7270/Q2KW5K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transitional endoplasmic reticulum ATPase (Homo sapiens (Human)) | BDBM50500324![]() (CHEMBL3747448) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Cleave Biosciences Inc. Curated by ChEMBL | Assay Description Inhibition of p97 ATPase in human A549 cells assessed as reduction in p62 protein incubated for 6 hrs by immunofluorescence assay | J Med Chem 58: 9480-97 (2015) Article DOI: 10.1021/acs.jmedchem.5b01346 BindingDB Entry DOI: 10.7270/Q2KW5K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transitional endoplasmic reticulum ATPase (Homo sapiens (Human)) | BDBM50500324![]() (CHEMBL3747448) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Cleave Biosciences Inc. Curated by ChEMBL | Assay Description Inhibition of p97 ATPase in human A549 cells assessed as accumulation of K48 poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence as... | J Med Chem 58: 9480-97 (2015) Article DOI: 10.1021/acs.jmedchem.5b01346 BindingDB Entry DOI: 10.7270/Q2KW5K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transitional endoplasmic reticulum ATPase (Homo sapiens (Human)) | BDBM50500324![]() (CHEMBL3747448) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 580 | n/a | n/a | n/a | n/a | n/a | n/a |
Cleave Biosciences Inc. Curated by ChEMBL | Assay Description Inhibition of p97 ATPase in human A549 cells assessed as accumulation of CHOP poly-ubiquitinated proteins incubated for 6 hrs by immunofluorescence a... | J Med Chem 58: 9480-97 (2015) Article DOI: 10.1021/acs.jmedchem.5b01346 BindingDB Entry DOI: 10.7270/Q2KW5K2P | |||||||||||
More data for this Ligand-Target Pair |