Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Transmembrane prolyl 4-hydroxylase' and Ligand = 'BDBM109267'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human))	BDBM109267 (US8609698, 8) Show SMILES Cc1ccnc(c1)-n1[nH]cc(-c2cncc(c2)C#N)c1=O Show InChI InChI=1S/C15H11N5O/c1-10-2-3-18-14(4-10)20-15(21)13(9-19-20)12-5-11(6-16)7-17-8-12/h2-5,7-9,19H,1H3	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	5.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Bayer Intellectual Property GmbH US Patent					Assay Description Inhibition of the Activity of HIF Prolyl Hydroxylase is carried out as described [Oehme F., Jonghaus W., Narouz-Ott L., Huetter J., Flamme I., Anal. ...				US Patent US8609698 (2013) BindingDB Entry DOI: 10.7270/Q2G44NZ8
					More data for this Ligand-Target Pair