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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase receptor UFO' and Ligand = 'BDBM531965'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Tyrosine-protein kinase receptor UFO


(Homo sapiens (Human))
BDBM531965
PNG
(US11208403, Example 42)
Show SMILES COc1ccnc(N)c1-c1ccc(NC(=O)c2cn(CC3CCOCC3)cc(-c3ccc(C)cc3)c2=O)cc1F |(9.34,-.77,;8,-1.54,;8,-3.08,;9.34,-3.85,;9.34,-5.39,;8,-6.16,;6.67,-5.39,;5.33,-6.16,;6.67,-3.85,;5.33,-3.08,;4,-3.85,;2.67,-3.08,;2.67,-1.54,;1.33,-.77,;,-1.54,;,-3.08,;-1.33,-.77,;-1.33,.77,;-2.67,1.54,;-2.67,3.08,;-1.33,3.85,;,3.08,;1.33,3.85,;1.33,5.39,;,6.16,;-1.33,5.39,;-4,.77,;-4,-.77,;-5.33,-1.54,;-6.67,-.77,;-8,-1.54,;-8,-3.08,;-9.34,-3.85,;-6.67,-3.85,;-5.33,-3.08,;-2.67,-1.54,;-2.67,-3.08,;4,-.77,;5.33,-1.54,;6.67,-.77,)|
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 1.30n/an/an/an/an/an/a


TBA

Assay Description
A kinase dilution solution containing 170 ng/ml AXL (the 464th to 885th amino acids of the intracellular domain of human AXL expressed as a fusion pr...


Citation and Details

BindingDB Entry DOI: 10.7270/Q29026Z6
More data for this
Ligand-Target Pair