Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vitamin D3 receptor (Rattus norvegicus) | BDBM50417514 (CHEMBL1630754) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Displacement of [3H]1alpha,25-(OH)2D3 from rat recombinant full length VDR | J Med Chem 53: 8642-9 (2010) Article DOI: 10.1021/jm1010447 BindingDB Entry DOI: 10.7270/Q23B61D2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vitamin D3 receptor (Rattus norvegicus) | BDBM50417514 (CHEMBL1630754) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Wisconsin-Madison Curated by ChEMBL | Assay Description Activity at rat recombinant full length VDR expressed in rat ROS 17/2.8 cells transfected with 24-hydroxylase gene promoter assessed as transcription... | J Med Chem 53: 8642-9 (2010) Article DOI: 10.1021/jm1010447 BindingDB Entry DOI: 10.7270/Q23B61D2 | |||||||||||
More data for this Ligand-Target Pair |