Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427129![]() (CHEMBL2323441) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427127![]() (CHEMBL2323442) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427131![]() (CHEMBL2323446) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427125![]() (CHEMBL2323444) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427130![]() (CHEMBL2323447) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427126![]() (CHEMBL2323443) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427124![]() (CHEMBL2323445) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (RAT) | BDBM50427128![]() (CHEMBL2321893) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shanghai Jiao Tong University School of Medicine Curated by ChEMBL | Assay Description Displacement of [3H]NMS from muscarinic M2 receptor in Sprague-Dawley rat left atria after 60 mins | Bioorg Med Chem 21: 1234-9 (2013) Article DOI: 10.1016/j.bmc.2012.12.052 BindingDB Entry DOI: 10.7270/Q2DF6SHB | |||||||||||
More data for this Ligand-Target Pair |