Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50003015 (CHEMBL227378) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.54E+4 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human muscarinic M2 receptor expressed in CHO cells | Bioorg Med Chem 15: 886-96 (2007) Article DOI: 10.1016/j.bmc.2006.10.040 BindingDB Entry DOI: 10.7270/Q2930WX9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50003015 (CHEMBL227378) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.51E+4 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human muscarinic M4 receptor expressed in CHO cells | Bioorg Med Chem 15: 886-96 (2007) Article DOI: 10.1016/j.bmc.2006.10.040 BindingDB Entry DOI: 10.7270/Q2930WX9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50003015 (CHEMBL227378) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.01E+4 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human muscarinic M3 receptor expressed in CHO cells | Bioorg Med Chem 15: 886-96 (2007) Article DOI: 10.1016/j.bmc.2006.10.040 BindingDB Entry DOI: 10.7270/Q2930WX9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50003015 (CHEMBL227378) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.94E+5 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Agonist activity at human muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem 15: 886-96 (2007) Article DOI: 10.1016/j.bmc.2006.10.040 BindingDB Entry DOI: 10.7270/Q2930WX9 | |||||||||||
More data for this Ligand-Target Pair |