Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50169951 ((6aR,10aR)-3-Adamantan-1-yl-6,6,9-trimethyl-6a,7,1...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.53E+3 | n/a | n/a | n/a | n/a |
Northeastern University Curated by ChEMBL | Assay Description Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 mins | J Med Chem 56: 3904-21 (2013) Article DOI: 10.1021/jm4000775 BindingDB Entry DOI: 10.7270/Q2VQ3429 | |||||||||||
More data for this Ligand-Target Pair |