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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50206934   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucocorticoid receptor


(Homo sapiens (Human))		BDBM50206934
PNG
(CHEMBL3937005)
Show SMILES [H][C@@]12CC[C@@](O)(C#CCCCC)[C@@]1(C)C[C@H](O)[C@]1([H])c3ccc(cc3CC[C@@]21[H])C(=O)Nc1cccnc1C |r|
Show InChI InChI=1S/C31H38N2O3/c1-4-5-6-7-15-31(36)16-14-25-24-13-10-21-18-22(29(35)33-26-9-8-17-32-20(26)2)11-12-23(21)28(24)27(34)19-30(25,31)3/h8-9,11-12,17-18,24-25,27-28,34,36H,4-6,10,13-14,16,19H2,1-3H3,(H,33,35)/t24-,25-,27-,28+,30-,31-/m0/s1
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Article
PubMed
n/an/an/an/a 100n/an/an/an/a



The Scripps Research Institute

Curated by ChEMBL


Assay Description
Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...

Bioorg Med Chem Lett 27: 347-353 (2017)


Article DOI: 10.1016/j.bmcl.2016.11.007
BindingDB Entry DOI: 10.7270/Q24B339Q
More data for this
Ligand-Target Pair