Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Muscarinic acetylcholine receptor M4 (RAT) | BDBM50249030 (CHEMBL3770346) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 225 | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Positive allosteric modulation of rat M4 receptor expressed in CHO cells co-expressing Gqi5 assessed as increase in acetylcholine-induced calcium mob... | Bioorg Med Chem Lett 27: 4999-5001 (2017) Article DOI: 10.1016/j.bmcl.2017.10.016 BindingDB Entry DOI: 10.7270/Q2SJ1P6M | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |