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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 153400   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Phosphodiesterase


(Trypanosoma brucei)		BDBM153400
PNG
(4-((3-Methoxyphenyl)amino)-8-methyl-6-(3-morpholin...)
Show SMILES COc1cccc(Nc2c(cnc3c(C)cc(cc23)-c2cccc(c2)N2CCOCC2)C(N)=O)c1
Show InChI InChI=1S/C28H28N4O3/c1-18-13-20(19-5-3-7-22(14-19)32-9-11-35-12-10-32)15-24-26(18)30-17-25(28(29)33)27(24)31-21-6-4-8-23(16-21)34-2/h3-8,13-17H,9-12H2,1-2H3,(H2,29,33)(H,30,31)
PDB

UniProtKB/TrEMBL

B.MOAD
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/a 1.20E+4n/an/an/an/a7.4n/a



Northeastern University



Assay Description
In short, recombinant TbrPDEB1 and TbrPDEB2 were assayed in 10 mM Tris pH 7.4, bovine serum albumin (0.2 mg/mL), 10 mM MgCl2, 25µM cAMP (Enzo Lifesci...

Chem Biol Drug Des 85: 549-64 (2015)


Article DOI: 10.1111/cbdd.12443
BindingDB Entry DOI: 10.7270/Q2FF3R28
More data for this
Ligand-Target Pair