Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 8 (Homo sapiens (Human)) | BDBM50004051 (2-Amino-4-phosphono-butyric acid | 2-Amino-4-phosp...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Inhibitory concentration against [3H]1 binding to recombinant human Metabotropic glutamate receptor 8 | Bioorg Med Chem Lett 15: 349-51 (2004) Article DOI: 10.1016/j.bmcl.2004.10.093 BindingDB Entry DOI: 10.7270/Q2G161M2 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamine--fructose-6-phosphate aminotransferase [isomerizing] (Candida albicans) | BDBM50004051 (2-Amino-4-phosphono-butyric acid | 2-Amino-4-phosp...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | 1.20E+7 | n/a | 2.60E+7 | n/a | n/a | n/a | n/a | 6.85 | n/a | |
Technical University of Gdansk | Assay Description Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua... | Bioorg Chem 25: 283-296 (1997) BindingDB Entry DOI: 10.7270/Q2RB7351 | |||||||||||
More data for this Ligand-Target Pair |