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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50090435   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein c-Fos/Transcription factor Jun


(Homo sapiens (Human))		BDBM50090435
PNG
(3-Methyl-1-[5-(3-methyl-isoxazol-5-yl)-2-thiophen-...)
Show SMILES CC1=CC(=O)N(Nc2nc(ncc2-c2cc(C)no2)-c2cccs2)C1=O |t:1|
Show InChI InChI=1S/C17H13N5O3S/c1-9-6-14(23)22(17(9)24)20-15-11(12-7-10(2)21-25-12)8-18-16(19-15)13-4-3-5-26-13/h3-8H,1-2H3,(H,18,19,20)
PDB

KEGG

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
PubMed
n/an/a 300n/an/an/an/an/an/a



Signal Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cells

Bioorg Med Chem Lett 10: 1645-8 (2000)


BindingDB Entry DOI: 10.7270/Q2F190XH
More data for this
Ligand-Target Pair