Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein phosphatase 2A activator (Homo sapiens (Human)) | BDBM50127375 ((E)-(R)-4-Hydroxy-2-methyl-hex-2-enedioic acid 6-{...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California at Irvine Curated by ChEMBL | Assay Description Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assay | Bioorg Med Chem Lett 13: 1597-600 (2003) BindingDB Entry DOI: 10.7270/Q2DB82CK | |||||||||||
More data for this Ligand-Target Pair |