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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50187207   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histone-lysine N-methyltransferase SETD7


(Homo sapiens (Human))		BDBM50187207
PNG
(CHEMBL3827431)
Show SMILES CN1CCC(CC1)OC1c2ccccc2Sc2ccccc12
Show InChI InChI=1S/C19H21NOS/c1-20-12-10-14(11-13-20)21-19-15-6-2-4-8-17(15)22-18-9-5-3-7-16(18)19/h2-9,14,19H,10-13H2,1H3
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Article
PubMed
n/an/a>1.00E+5n/an/an/an/an/an/a



Tokyo Medical and Dental University (TMDU)

Curated by ChEMBL


Assay Description
Inhibition of recombinant SET7/9 (unknown origin) using biotinylated histone H3-derived peptide/SAM as substrate after 60 mins by AlphaLISA assay

Bioorg Med Chem 24: 4318-4323 (2016)


Article DOI: 10.1016/j.bmc.2016.07.024
BindingDB Entry DOI: 10.7270/Q2959KGV
More data for this
Ligand-Target Pair