Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50201275 (7-fluoro-4-oxo-N-(1-(3-oxo-2,3,4,6,7,8-hexahydroin...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description Displacement of 125I-MCH from MCH-R1 expressed in IMR-32 cells | Bioorg Med Chem Lett 17: 884-9 (2007) Article DOI: 10.1016/j.bmcl.2006.11.061 BindingDB Entry DOI: 10.7270/Q2J38S6V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50201275 (7-fluoro-4-oxo-N-(1-(3-oxo-2,3,4,6,7,8-hexahydroin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.46E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description Displacement of 3H-dofetilide from hERG-expressing HEK membrane homogenates | Bioorg Med Chem Lett 17: 884-9 (2007) Article DOI: 10.1016/j.bmcl.2006.11.061 BindingDB Entry DOI: 10.7270/Q2J38S6V | |||||||||||
More data for this Ligand-Target Pair |