Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcription factor Jun (Homo sapiens (Human)) | BDBM50213936 ((S)-2,3,6,7-tetramethoxy-8b,9,10,11,12,12a-hexahyd...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >300 | n/a | n/a | n/a | n/a | n/a | n/a |
Yale University Curated by ChEMBL | Assay Description Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assay | Bioorg Med Chem Lett 17: 4338-42 (2007) Article DOI: 10.1016/j.bmcl.2007.05.021 BindingDB Entry DOI: 10.7270/Q2HD7VBW | |||||||||||
More data for this Ligand-Target Pair |